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2-methyl-5-{4-[(3-methylthiophen-2-yl)sulfonyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
2-{3-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
N-(1,5-dimethyl-1H-pyrazol-4-yl)-2-[3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]acetamide
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
6-[3-(1,3-benzoxazol-2-yl)piperidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-1H-imidazole
N-(3-phenylpropyl)-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
(2S,4R)-4-amino-N-methyl-1-{5-[(4-methylpiperidin-1-yl)methyl]furan-2-carbonyl}pyrrolidine-2-carboxamide
methyl (2S,4R)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-(quinolin-4-ylmethyl)pyrrolidine-2-carboxylate
5-{2-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(cyclopropylmethyl)-1-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-[4-({[(1-methylpiperidin-3-yl)methyl](2-phenylethyl)amino}methyl)thiophen-2-yl]ethan-1-one
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidine-4-carboxamide
7-(5-chloropyridin-2-yl)-4-[(2R)-oxolane-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1R,2S)-2-[2-(2-ethoxyphenyl)-1H-imidazol-1-yl]cyclopentan-1-ol
7-[(2-fluorophenyl)methyl]-2-(pyrimidin-2-yl)-2,7-diazaspiro[4.5]decane
2-{5-[(3-acetyl-7-ethyl-1H-indol-1-yl)methyl]-3-cyclopropyl-1H-1,2,4-triazol-1-yl}acetic acid
4-[(2,6-difluoro-3-methoxyphenyl)methyl]-1-(2-phenylethyl)piperazin-2-one
1-(carbamoylmethyl)-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-methyl-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
3-({[2-(diethylamino)pyridin-3-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
2-(pyridin-2-ylmethyl)-9-(4,4,4-trifluorobutanoyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
(2S,4R)-4-amino-N-ethyl-1-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]pyrrolidine-2-carboxamide
N,N-dimethyl-3-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]aniline
4-[(dimethylamino)methyl]-1-(2,5,7-trimethylquinoline-4-carbonyl)azepan-4-ol
5-fluoro-N-methyl-2-(2-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)pyrimidin-4-amine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-5-(methoxymethyl)-N-methylfuran-2-carboxamide
3-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl](methyl)amino}-N-methylpropanamide
(2R,3R)-1'-(1H-pyrazole-3-carbonyl)-3-(1,2,3,6-tetrahydropyridin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-(carbamoylmethyl)-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}piperidine-3-carboxamide
2-ethyl-7-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
1-[2-(1,4-oxazepan-4-ylmethyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
3-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methoxyphenyl]-N,N,1-trimethyl-1H-1,2,4-triazol-5-amine
1-(2-{[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}ethyl)-4,6-dimethyl-1,2-dihydropyrimidin-2-one
[(1-ethyl-1H-indol-4-yl)methyl](methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
(1R,5S,6R)-3-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
methyl 4-({2-[(3-chlorophenyl)methyl]-1,3-benzoxazol-6-yl}formamido)butanoate
{2-[3-(2-ethylphenoxy)azetidin-1-yl]-8-methylquinolin-3-yl}methanol
2-(3-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propane-1,3-diol
1-[(5-ethylfuran-2-yl)methyl]-3-(pyrrolidin-1-yl)piperidine
1-methyl-3-(2-methylpropyl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]-1H-pyrazole-5-carboxamide
7-(4-chlorophenyl)-2-[2-(diethylamino)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-(piperidine-1-carbonyl)piperidine
1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]acetamide
2-methoxy-N-[2-methyl-3-({[3-(oxolan-3-yl)propyl]carbamoyl}amino)phenyl]acetamide
[(3R,4R)-1-(2-methyl-1,3-benzothiazole-5-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-[3-(1H-indol-2-yl)phenyl]-1-[(6-methylpyridin-2-yl)methyl]piperidine-3-carboxamide