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N-[(5-fluoro-2-methylphenyl)methyl]-5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carboxamide
1-{[(3-methyl-1-propyl-1H-pyrazol-4-yl)formamido]methyl}cyclopentane-1-carboxylic acid
N-[3-(dimethylamino)propyl]-1-(2,5-dimethylbenzenesulfonyl)-N-methylpiperidin-3-amine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
N-cyclobutyl-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
6-(4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)-1H-indole
2-({[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
2-[4-(2H-1,3-benzodioxol-4-ylmethyl)-1-[(4-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-3-methanesulfonylpropan-1-one
2-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}-2,7-diazaspiro[4.5]decan-6-one
3-(oxolan-3-yl)-5-[4-(pyrrolidin-1-ylmethyl)phenyl]-1,2,4-oxadiazole
(1S,5R)-6-benzyl-3-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(3-fluorophenyl)methyl]-4-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}piperazine
3-{1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}pyridine
1-(2-methanesulfonylethyl)-4-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]piperazine
4-(hydroxymethyl)-1-(2-methoxy-5-methylbenzenesulfonyl)azepan-4-ol
5-ethyl-N-[(3S)-2-oxoazepan-3-yl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
(2E)-N-({3-methyl-7-[4-(1H-pyrazol-1-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
(1S,5R)-6-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
6-(furan-3-yl)-2-(4-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}phenyl)-3,4-dihydropyrimidin-4-one
1-(dimethylsulfamoyl)-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
[(3R,4R)-1-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
2-(5-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}furan-2-yl)benzonitrile
1-[(4aR,8aS)-1-{imidazo[1,2-a]pyridine-2-carbonyl}-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
2-({5-[2-(2-hydroxyphenyl)ethyl]-4-(pyridin-3-yl)-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
3-[3-(3-methylpyridin-2-yl)-1,2,4-oxadiazol-5-yl]-4,5,6,7-tetrahydro-2H-indazole
3-[3-(3-chlorophenyl)pyrrolidin-1-yl]-5-(4-methoxyphenyl)-1,2,4-triazine
1-[(4-hydroxyphenyl)methyl]-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
3-{2-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
3-[2-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-1,3-oxazolidin-2-one
2-[3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methylpropanamido]acetic acid
5-{[(5-methyl-1H-pyrazol-3-yl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(3E)-1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]pent-3-en-1-one
1-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-N-[3-(oxolan-3-yl)propyl]piperidin-4-amine
N-(2-methoxyethyl)-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
1-[2-(3-chlorophenyl)ethyl]-4-[(dimethylsulfamoyl)amino]pyrrolidin-2-one
(3S,4R)-1-(5-chloro-3-fluoropyridin-2-yl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
6-(furan-3-yl)-2-[3-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
6-(4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)pyridine-3-carboxylic acid
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(piperidin-1-yl)ethyl]acetamide
(3S,4R)-4-(pyridin-4-yl)-1-(quinoxaline-6-carbonyl)pyrrolidine-3-carboxylic acid
2-{[4-(3-chlorophenyl)-5-[(4-hydroxyphenyl)methyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-[(6-amino-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)amino]-N-cyclopropylacetamide
2-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-N-(thiophen-2-ylmethyl)acetamide
methyl 2-{1-[(2E)-2-methylbut-2-en-1-yl]-3-oxopiperazin-2-yl}acetate
4-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-N,N,6-trimethylpyrimidin-2-amine
1-{4-[3-(4H-1,2,4-triazol-4-yl)phenyl]phenyl}piperazine
6-cyclobutyl-2-(3-{[3-(trifluoromethyl)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
1-(2-aminoethyl)-N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide