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5-chloro-3-[3-(furan-2-yl)-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]-4,6-dimethyl-1,2-dihydropyridin-2-one
1-(prop-2-en-1-yl)-5-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-methyl-4-(5-methylfuran-2-yl)-N-(piperidin-4-yl)benzamide
N-{[2-(dimethylamino)-7-(methylsulfanyl)quinolin-3-yl]methyl}-2-ethyl-N-(furan-2-ylmethyl)butanamide
1-{3-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(1H-indol-2-ylmethyl)-1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]piperidin-4-amine
2-acetyl-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
3-{1-[1-(2-hydroxyethyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]ethyl}-3,4-dihydroquinazolin-4-one
4-(3,3-diphenylpiperidine-1-carbonyl)pyrrolidin-2-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-4-methyl-N-(oxolan-2-ylmethyl)-1,2,5-oxadiazole-3-carboxamide
2-(azepan-1-yl)-N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]acetamide
2,3-dimethyl-7-{6-methylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
2-{[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}benzoic acid
5-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-[(3S,5S)-1-ethyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1-methyl-5-phenyl-1H-pyrrole-2-carboxamide
methyl 3-chloro-4-({[2-(1-methylpyrrolidin-2-yl)ethyl]carbamoyl}amino)benzoate
1-(1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)-3-phenylpropan-1-one
2-[2-(1,2-benzoxazol-3-yl)acetamido]-N-(2-fluoro-4-methylphenyl)propanamide
(3-{2-[1-(3,4-difluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-{2-[(2R,6R)-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}ethan-1-one
3-{[(2-methoxyethyl)[(4-methylphenyl)methyl]amino]methyl}-N-methylpyridin-2-amine
dimethyl({[(3S,4R)-1-(2-phenylethyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl})amine
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
7-chloro-2-methyl-4-{1-oxa-7-azaspiro[3.5]nonane-7-carbonyl}quinoline
2,5-dimethyl-N-[3-(methylsulfanyl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
8-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decane
2-[(3S,7S)-3-(hydroxymethyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-trien-5-yl]-6-methylpyridine-3-carbonitrile
methyl 5-[4-(2-{[(3-chlorophenyl)methyl]carbamoyl}ethyl)piperidin-1-yl]-5-oxopentanoate
4-[2-(4-methyl-1H-pyrazol-1-yl)propanoyl]-1-(4-methylphenyl)piperazin-2-one
5-benzyl-N-[1-(furan-2-yl)ethyl]-N-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-(4-fluorophenyl)-1-(5-fluoroquinazolin-4-yl)piperidin-4-ol
4-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}pyrrolidin-2-yl)-3,5-dimethyl-1,2-oxazole
(2R,4S)-4-hydroxy-1-{[1-(propan-2-yl)piperidin-4-yl]methyl}piperidine-2-carboxylic acid
1-[2-(2-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-4-oxo-N-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
5-(2H-1,3-benzodioxol-5-yl)-2-chloro-N-methylbenzamide
1-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-2-(4,6,7-trimethyl-1-benzofuran-3-yl)ethan-1-one
8-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-carbonyl}-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
4-hydroxy-2-(phenoxymethyl)-N-[2-(1,3-thiazol-4-yl)ethyl]pyrimidine-5-carboxamide
N-[2-(4-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-4-yl}-1,2,3,6-tetrahydropyridin-1-yl)ethyl]acetamide
N-[2-(4-fluorobenzenesulfonyl)ethyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
(2-methoxyethyl)[2-phenyl-1-(1-propylpiperidin-4-yl)ethyl](pyridin-3-ylmethyl)amine
4-[3-(2H-1,3-benzodioxol-5-ylmethyl)-1,2,4-oxadiazol-5-yl]-2-methoxyphenol
N-{1-[(2-fluorophenyl)methyl]azepan-4-yl}-2-(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)acetamide
7-[(2-aminopyridin-3-yl)methyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
ethyl 4-[(2-chlorophenyl)methyl]-1-[2-(methylsulfanyl)acetyl]piperidine-4-carboxylate
2-(cyclopropylmethyl)-9-[(5-fluoro-2-methoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
benzyl(oxolan-2-ylmethyl){[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
N-(oxolan-2-ylmethyl)-3-(pyridin-3-yl)-N-(thiophen-3-ylmethyl)propanamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide