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N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)acetamide
(3S,7S)-5-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]-N-[(3,4-difluorophenyl)methyl]propanamide
7-fluoro-N-[2-(7-methyl-1H-indol-3-yl)ethyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
5-{1-cyclopentyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1,3-dimethyl-1H-pyrazole
N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
3-[5-({[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amino}methyl)thiophen-3-yl]prop-2-yn-1-ol
[4-(4-cyclopentylpyrimidin-2-yl)morpholin-2-yl]methanamine
N-(3,4-difluorophenyl)-5-[4-hydroxy-1-(2-methylpropyl)piperidin-4-yl]-1-benzofuran-2-carboxamide
4-{1-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetamide
5-(3-chloro-2-fluorobenzoyl)-1-methyl-N-[2-(morpholin-4-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[3-(4-methyl-1,3-thiazol-5-yl)propyl]({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine
3-(2-methoxyphenyl)-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)propanamide
4-(2-{[5-(piperidin-1-ylmethyl)pyridin-2-yl]oxy}hex-5-en-1-yl)morpholine
N-{1-[(2-cyclohexylpyrimidin-5-yl)methyl]piperidin-4-yl}methanesulfonamide
N-{[1-(ethoxymethyl)cyclopropyl]methyl}-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
2-[4-phenyl-1-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1H-imidazol-5-yl]quinoline
1-({3-[(dimethylamino)methyl]phenyl}methyl)-1-methyl-3-(5-methyl-1,3,4-thiadiazol-2-yl)urea
1-benzoyl-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-cyclobutanecarbonyl-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}piperidine
(1S,5R)-3-[(5-methylfuran-2-yl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-(4-methyl-2-oxo-1,2-dihydroquinolin-7-yl)-3-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}urea
2-[(5-{[(3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl)amino]methyl}pyrimidin-2-yl)amino]acetic acid
N-(2-methoxyethyl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
4-({[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}methyl)-N-methylbenzene-1-sulfonamide
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-[3-(4-methyl-1,3-thiazol-2-yl)propyl]urea
3-(2-chlorophenyl)-1-methyl-6-(thiolan-3-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-{3-[(3-hydroxyazetidin-1-yl)methyl]-6-methylquinolin-2-yl}piperidin-3-ol
1-(2-amino-4-phenylpyrimidine-5-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
(3S)-3-ethyl-4-[(2-ethyl-1,3-thiazol-4-yl)methyl]morpholine
1-(2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)-3,3-dimethylurea
methyl[(6-methylpyridin-2-yl)methyl](quinolin-3-ylmethyl)amine
(3S,4S)-4-[(6-methyl-2-propylpyrimidin-4-yl)amino]-1-(propan-2-yl)pyrrolidin-3-ol
N-[(3,4-dimethoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)-4-(1H-1,2,4-triazol-1-yl)butanamide
8-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
5-(3-{1-[(4-methoxypyridin-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
4-(3-chloropyridin-2-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(1,2-oxazol-5-ylmethyl)acetamide
4-({4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
N-[1-({1-[(2E)-but-2-en-1-yl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)piperidin-4-yl]-2-methoxyacetamide
(2S,4R)-4-amino-N-ethyl-1-(5-phenyl-1H-pyrrole-2-carbonyl)pyrrolidine-2-carboxamide
5-(3-chloro-4-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-5-propyl-1,3,4-oxadiazol-2-amine
6-(4-cyclohexylpiperazine-1-carbonyl)-2-cyclopropyl-1,3-benzoxazole
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-[(4-chloro-3-fluorophenyl)methyl]piperazin-2-one
N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethyl-4-(hydroxymethyl)benzamide
3-(4-acetyl-4-phenylpiperidine-1-carbonyl)benzonitrile
8-(butan-2-yl)-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{4-[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1,4-diazepan-1-yl}ethan-1-one