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2,8-dimethyl-4-(2-phenylmorpholine-4-carbonyl)quinoline
3-[2-(azocan-1-yl)-2-oxoethyl]-4-(2,3-dihydro-1H-inden-2-yl)piperazin-2-one
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{2-[(4-fluorophenyl)formamido]ethyl}propanamide
3-{[(1-cyclobutylethyl)amino]methyl}-2-methoxy-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
(3aR,6aS)-5-[3-(2-methyl-1H-indol-1-yl)propanoyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-[(2-chloro-5-fluorophenyl)methyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{[4-(quinolin-4-yl)-1H-1,2,3-triazol-1-yl]methyl}-1λ6-thiolane-1,1-dione
1-{imidazo[1,2-b]pyridazin-6-yl}-4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperazine
(2E)-2-methyl-1-{3-[4-(naphthalen-1-yl)-1H-pyrazol-5-yl]piperidin-1-yl}but-2-en-1-one
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-[(1-propyl-1H-imidazol-2-yl)methyl]-1,4-diazepane
5-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
1-[(6-chloro-2H-chromen-3-yl)methyl]-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
5-[2-(aminomethyl)morpholine-4-carbonyl]-1,3-benzothiazol-2-amine
3-(4-hydroxyphenyl)-2-phenyl-N-[(1s,4s)-4-aminocyclohexyl]propanamide
4-{1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazol-2-yl}-2,1,3-benzoxadiazole
ethyl 1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
3-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
(4aR,8aS)-1-butyl-6-(1-methylpiperidin-4-yl)-decahydro-1,6-naphthyridin-2-one
3-{5-[2-(1H-indol-3-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
1-(cyclopropanesulfonyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
methyl 4-(4-{[benzyl(2-hydroxyethyl)amino]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
4-{[1-(2-methoxyphenyl)-5-(4-methyl-1,3-oxazol-5-yl)-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
2-methyl-3-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)quinoxaline
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-methyl-N-(1-methylpyrrolidin-3-yl)-1,2-oxazole-3-carboxamide
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-3-yl]-N-(2-hydroxyethyl)propanamide
4-(quinoline-6-carbonyl)-7-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5,6-dimethyl-2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-1,3-benzodiazole
8-[3-(1H-imidazol-1-yl)propyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-7-fluoro-1-(pyridin-3-ylmethyl)-1,2-dihydroquinolin-2-one
2-(prop-2-ene-1-sulfonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
{[4-(3-chlorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]methyl}[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
N-cyclopentyl-4-(4-{[1-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]amino}piperidin-1-yl)benzamide
1-[(3-methylphenyl)methyl]-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aR,7aS)-N-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-2-(phenylamino)pyrimidine-5-carboxamide
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methylpyrrolidine-3-carboxamide
2-[methyl(phenyl)amino]-1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-(2-methoxyethyl)-8-(2-methylpropyl)-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-methylpiperidin-1-yl)-N-{[1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]methyl}acetamide
3-methyl-7-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-ethyl-6-(1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
1-[4-fluoro-2-(1H-imidazol-2-yl)phenyl]-3,5-dimethyl-1H-pyrazole
N-{[5-({cyclopropyl[(2-methoxyphenyl)methyl]amino}methyl)furan-2-yl]methyl}-N-methylmethanesulfonamide
(isoquinolin-5-ylmethyl)(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-benzyl-3-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-N-methylpropanamide
8-(2-ethylpyridine-4-carbonyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2H-1,3-benzodioxole-5-carbonyl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid