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8-(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)-2H,5H,6H,7H,8H-[1,3]dioxolo[4,5-g]quinolin-6-one
4-(4-chloro-1-ethyl-1H-pyrazole-5-carbonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
1-ethyl-N-[2-(methylsulfanyl)ethyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
[3-(2-methylpropyl)-1-(5-propyl-1,3,4-oxadiazole-2-carbonyl)piperidin-3-yl]methanol
2-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4H-chromen-4-one
4-[(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}phenyl)methyl]morpholine
{4-[(3-methoxyphenyl)methyl]-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}methanol
4-{[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}quinoline
1-methyl-3-{[2-methyl-4-(2-methylphenyl)-5-oxopiperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
4-chloro-N-(1H-imidazol-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2,6-dimethylquinoline-3-carboxamide
5-fluoro-N,1,3-trimethyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H-indole-2-carboxamide
4-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-6-methylpyrimidine
3-(1-ethyl-1H-1,2,4-triazol-3-yl)-1-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}urea
4-(2-chloro-6-methoxyphenyl)-2-methyl-1H-imidazole
(2R,6R)-4-[(4-fluoro-3-methoxyphenyl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-{5-[2-(2-ethoxyethoxy)phenyl]-1,2,4-oxadiazol-3-yl}pyridazine
ethyl({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}){[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-({[1-(2,3-difluoro-6-methoxybenzoyl)piperidin-4-yl]oxy}methyl)pyridine
1-[3-(6-methylpyridin-2-yl)phenyl]ethan-1-one
3-(5-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}furan-2-yl)-1H-pyrazole
1-(2-methylpropyl)-4-(4-phenyl-5-propyl-1H-imidazol-2-yl)pyrrolidin-2-one
1-[(3-fluorophenyl)methyl]-4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]-1,4-diazepane
5-{[4-(oxan-4-yl)piperazin-1-yl]methyl}-2-(pyrrolidin-1-yl)pyrimidine
4-(6-methylpyridine-3-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{2-[1-(3-fluorophenyl)-1H-1,2,4-triazol-5-yl]phenyl}morpholine
(1R,5R)-3-(benzenesulfonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonane
4-[(2-chloro-6-fluorophenyl)methyl]-3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]piperazin-2-one
N-[(4-chlorophenyl)methyl]-4-(4-methoxyphenyl)-3-oxopiperazine-1-carboxamide
methyl 7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-3-{spiro[2.5]octane-1-carbonyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(1-methyl-1H-pyrazol-4-yl)-1-{spiro[indene-1,4'-piperidine]-1'-yl}propan-1-one
1-(2-benzyl-1,3-thiazole-4-carbonyl)-3-(1-ethyl-1H-imidazol-2-yl)piperidine
(3S,4R)-1-[2-(methylamino)-1,3-thiazole-4-carbonyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-ethyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1H-pyrazole-4-carboxamide
1-{4-[1-(1-methylpiperidin-4-yl)-3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]thiophen-2-yl}ethan-1-one
4-{1-[1-(ethanesulfonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
4-[3-(4-cyclopentyl-1,4-diazepane-1-carbonyl)phenyl]-2-methylbutan-2-ol
3-({[(2,2-dimethyloxan-4-yl)methyl]amino}methyl)-N,N-dimethylpyridin-2-amine
1-[3-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
4-methoxy-6-(6-methylpyridin-3-yl)pyrimidin-2-amine
4-methyl-5-[2-(piperidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1,3-thiazol-2-amine
2-(2,2-dimethylpropanamido)-N-[(3-ethoxy-4-methoxyphenyl)methyl]-N,5-dimethylthiophene-3-carboxamide
5-chloro-3-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,2-dihydropyridin-2-one
N-[(2-ethoxy-3-methoxyphenyl)methyl]-N,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-(2-fluoro-4-methoxyphenyl)-2-methyl-4-[(4-methylphenyl)methyl]-3-oxopiperazine-1-carboxamide
3-[(4aR,7aS)-4-(2-hydroxybenzoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
(4aS,8aR)-1-(3-aminopropyl)-6-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(thiophen-2-yl)propan-1-one
3-(1H-1,3-benzodiazol-1-yl)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]propan-1-one
1-[cyclohexyl(methyl)amino]-3-{2-[(4,4-difluoropiperidin-1-yl)methyl]phenoxy}propan-2-ol