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(1-methyl-1H-imidazol-2-yl)({1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperidin-4-yl})methanol
1-[3-(4-phenylbenzoyl)piperidin-1-yl]pent-4-en-1-one
(1R,7S)-3-(2,2-dimethylpropyl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-(propan-2-yl)-5-{1-[3-(pyridin-3-yl)propyl]-1H-imidazol-2-yl}pyrimidine
6-fluoro-2-oxo-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-[(2-fluorophenyl)methyl]-3-(1-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}piperidin-3-yl)propanamide
4-[4-methoxy-3-(prop-2-en-1-yl)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-fluoro-2-methylphenyl)urea
3,4-difluoro-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-1,4-diazepan-6-ol
9-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}-4-methyl-1,4-diazepane
[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl){[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amine
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-hydroxy-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-(1H-imidazol-2-yl)-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)piperidine
methyl 3-[(2,2-dimethylpropanamido)methyl]-5-[2-(1H-pyrazol-1-yl)acetamido]benzoate
N-(1H-imidazol-2-ylmethyl)-N-methyl-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
(4aR,8aS)-6-[5-(4-methoxyphenyl)furan-2-carbonyl]-1-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
4-[(2,5-difluorophenyl)methyl]-7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-cycloheptyl-1-ethyl-N-[(3-methoxyphenyl)methyl]-1H-pyrazole-5-carboxamide
N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)pyrazine-2-carboxamide
1-[3-(3-methyl-2,5-dioxoimidazolidin-1-yl)phenyl]-3-[3-(pyrrolidin-1-yl)propyl]urea
(4aR,7aS)-1-(cyclopropylmethyl)-4-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(carbamoylmethyl)-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-(propan-2-yl)piperidine-3-carboxamide
4-(1-aminocyclopropanecarbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-{pyrazolo[1,5-a]pyridin-7-yl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{2-[1-(3-aminothiophene-2-carbonyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(5-methylthiophene-3-carbonyl)pyrrolidin-3-yl]methanol
[(1-cyclopentylpiperidin-4-yl)methyl][(5-methylthiophen-2-yl)methyl](oxolan-2-ylmethyl)amine
N-[1-(furan-2-yl)ethyl]-N-methyl-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
N-{[1-(morpholin-4-ylmethyl)cyclopropyl]methyl}-3-(pyridin-4-yl)propanamide
5-[3-(3-methoxypropyl)piperidine-1-carbonyl]pyridin-2-amine
(2,1,3-benzoxadiazol-4-ylmethyl)({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)amine
{4-[6-(piperidin-1-yl)pyrimidin-4-yl]phenyl}methanol
methyl 2-(1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
1-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-4-(thian-4-yl)piperazine
4-(4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-yl)pyridine
6-(4-methanesulfonylbenzoyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
8-(1,3-benzothiazol-2-ylmethyl)-1-benzyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1R,2R,6S,7S)-4-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-azatricyclo[5.2.1.02,6]decane
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
3-{3-ethyl-5-[2-(methylamino)pyridin-4-yl]-1H-1,2,4-triazol-1-yl}-4-fluorobenzene-1-sulfonamide
2-[4-(1,3-thiazol-2-ylmethyl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
5-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]pyrrolidin-2-yl}-N-phenylthiophene-2-carboxamide
N-[2-chloro-5-(2-methoxyacetamido)phenyl]-4,4-difluoropiperidine-1-carboxamide
5-cyclobutyl-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1,3,4-oxadiazol-2-amine
N-{[2-(methoxymethyl)-4-methyl-1,3-thiazol-5-yl]methyl}-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
2-methyl-1-({4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}methyl)-1,4-diazepan-5-one
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(furan-2-yl)-N-methyl-2-oxoacetamide
3-[2-(4-methoxyphenyl)ethyl]-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine