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N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-3-(1H-1,2,4-triazol-1-yl)propanamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)piperidin-2-one
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetamide
2-(4-{[4-(aminomethyl)piperidin-1-yl]methyl}phenyl)-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
N-[(3S,4R)-1-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
5-(2-chlorophenyl)-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]furan-2-carboxamide
2-{2-[2-(4-ethylphenyl)-1H-imidazol-1-yl]ethyl}pyrazine
1-[(4aR,8aR)-7-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
N,3-dimethyl-N-{2-[2-(prop-2-en-1-yl)phenoxy]ethyl}furan-2-carboxamide
2-[(6-methylpyridin-2-yl)methyl]-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
1'-[(5-methylfuran-2-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-{5-[1-(2H-1,3-benzodioxol-5-yloxy)ethyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
1-[(4-methoxyphenyl)methyl]-4-(1H-pyrrole-2-carbonyl)piperazin-2-one
6-oxo-7-(3-phenylpropyl)-N-(propan-2-yl)-2,7-diazaspiro[4.5]decane-2-carboxamide
2-butyl-N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1,3-benzoxazole-5-carboxamide
2-(6-methoxynaphthalen-2-yl)-4-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]morpholine
2-amino-4-[4-(2-hydroxyethoxy)phenyl]-6-(4-hydroxyphenyl)-5-methylpyridine-3-carbonitrile
N-[(2S)-1-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-4-methyl-1-oxopentan-2-yl]acetamide
4-[(3S,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]-1λ6-thiane-1,1-dione
5-{2-[(pyridin-3-ylmethyl)amino]ethyl}-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
4-[4-(methylamino)pyrimidin-2-yl]phenol
3-[5-(2-propyl-1,3-thiazol-4-yl)-1,2,4-oxadiazol-3-yl]pyridazine
4-[(2,4-difluorophenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[4-(cyclohexylmethyl)-1H-1,2,3-triazol-1-yl]piperidine
N1-(3-methylpyridin-2-yl)-N2-[4-(pyridin-4-yl)pyrimidin-2-yl]ethane-1,2-diamine
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carboxamide
(2R,6S)-4-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,6-dimethylmorpholine
N-(6-fluoropyridin-3-yl)-3-(1H-imidazol-1-ylmethyl)piperidine-1-carboxamide
N-cyclopentyl-N-[(5-methylthiophen-2-yl)methyl]pent-4-ynamide
1-(2-phenoxyethyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-(4-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-methyl-1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-2-phenylpiperazine
N-[3-(methylsulfanyl)propyl]-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-4-(4-methoxyphenyl)butan-1-one
N4-methyl-N2-[(1-methyl-4-phenylpiperidin-4-yl)methyl]pyrimidine-2,4-diamine
N-(1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
1-(oxolan-2-ylmethyl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N,2,4-trimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1,3-thiazole-5-carboxamide
4-[4-(3-chlorophenyl)-3-oxopiperazin-1-yl]-N-cyclopentyl-4-oxobutanamide
(3S,4R)-1-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-amino-6-(4-fluorophenyl)-4-(furan-3-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
5-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidine-1-carbonyl]pyridine-2-carbonitrile
(3S,4S)-1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(propan-2-yloxy)pyrrolidin-3-ol
3-[(2-fluorophenyl)formamido]-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]propanamide
2-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
2,5-dimethyl-3-[4-(1H-pyrazole-4-carbonyl)piperazin-1-yl]pyrazine
N-ethyl-4-[(3-methoxypropyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(trifluoromethyl)pyridine