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N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-7-fluoro-2-methylquinoline-4-carboxamide
4-({[(3-hydroxypiperidin-3-yl)methyl]amino}methyl)-1,2-dihydrophthalazin-1-one
3-{[9-cyclopentyl-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]methyl}phenol
(3S,9aR)-3-(4-aminobutyl)-8-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-[4-(4-ethylpiperazin-1-yl)piperidin-1-yl]-N-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-{[1-(1-methyl-1H-pyrazol-5-yl)propyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-(4-fluorophenyl)-1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-3-amine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(3-methylthiophen-2-yl)methyl]pyrrolidin-3-yl]pyridine-3-carboxamide
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-methyl-1,2-dihydroquinoxalin-2-one
1-ethyl-N-(furan-2-ylmethyl)-3-(2-methylpropyl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
6-(3-fluorophenyl)-N-[2-(pyridin-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(2-methoxy-5-methylphenyl)-5-methyl-1,3-benzoxazole
2-{2-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-6-methylpyridine-3-carbonitrile
(1S,5R)-6-(cyclopropylmethyl)-3-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propan-1-one
N-{[4-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-N-cyclopropylpyridine-3-carboxamide
2-methoxy-N-{[3-methyl-7-(2-methylfuran-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-phenylacetamide
N-(3-acetylphenyl)-2-[4-(2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)morpholin-3-yl]acetamide
({2-[(2-chlorophenyl)methoxy]-7-(methylsulfanyl)quinolin-3-yl}methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
3-cyclopentyl-6-[1-(propan-2-yloxy)ethyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
3-[5-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl){[1-(2-methylphenyl)-1H-1,2,3,4-tetrazol-5-yl](phenyl)methyl}amine
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(1-methyl-1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-benzyl-8-[6-(dimethylamino)pyrazin-2-yl]-2,8-diazaspiro[4.5]decan-3-one
N-(pyridin-3-yl)-3-[2-(pyrrolidin-1-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]propanamide
1-{4-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]phenyl}-2-(morpholin-4-yl)ethan-1-ol
2-(4-fluorophenyl)-N-(2-{7-[(3-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
6-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(5-methyl-1,3-oxazole-4-carbonyl)-4-(3-methylphenoxy)piperidine-4-carboxylic acid
2-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-1,3-benzothiazole
2-ethyl-N-(isoquinolin-5-ylmethyl)-N,4-dimethyl-1,3-oxazole-5-carboxamide
3-[(4-fluorophenyl)formamido]-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}propanamide
N-[3-(2-chlorophenoxy)propyl]-N-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2,7,8-trimethylquinoline-4-carboxamide
3,5-dimethyl-1-{1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]pyrrolidin-3-yl}-1H-pyrazole
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-(3-phenylpiperidin-1-yl)acetamide
(1S,5R)-3-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
dimethyl({[1-({1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methyl})amine
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(2-methyl-1-benzofuran-7-carbonyl)pyrrolidin-3-yl]methanol
4-[3-(2,3-dihydro-1H-indol-1-yl)propanoyl]-1-(4-methylphenyl)piperazin-2-one
2-({2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholin-4-yl}methyl)-4,5,6,7-tetrahydro-1,3-benzothiazole
1-cyclopentyl-5-oxo-N-{2-[4-(propan-2-yloxy)phenyl]ethyl}pyrrolidine-3-carboxamide
4,6-dimethyl-N-{1-oxaspiro[4.4]nonan-3-yl}-2-oxo-2H-pyran-5-carboxamide
4-[(benzyloxy)methyl]-3-propyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-methanesulfonyl-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)pyrrolidine-2-carboxamide
N-cyclopropyl-1-[(1s,4s)-4-{[(3-ethoxy-4-methoxyphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[3-(cyclohexyloxy)propyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
1-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(pyrimidin-2-ylsulfanyl)acetamide
N-(2-chloro-4-fluorophenyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide