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1-(3-chlorophenyl)-4-{1-[(2,5-dimethoxyphenyl)methyl]piperidin-3-yl}piperazine
(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methyl-N-[3-(methylsulfanyl)phenyl]piperidine-1-carboxamide
2-(4-cyclohexylpiperazin-1-yl)-2-[4-fluoro-3-(hydroxymethyl)phenyl]acetic acid
5-(methoxymethyl)-N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)furan-2-carboxamide
(1S,5R)-6-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
3-[2-(hydroxymethyl)phenyl]-5-(morpholine-4-sulfonyl)benzoic acid
2-amino-4-[4-ethoxy-3-(hydroxymethyl)phenyl]-6-(thiophen-2-yl)pyridine-3-carbonitrile
(3aR,6aR)-2-acetyl-5-({9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-phenylethyl)acetamide
4-(2-phenylpropyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(2-{[3-(dimethylsulfamoyl)-5-({[4-(2-methylpropyl)phenyl]methyl}amino)phenyl]formamido}ethyl)acetamide
1-cyclopentyl-4-{2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}piperazin-2-one
(3aS,6aS)-2-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-5-(1H-imidazol-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(1-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-1H-imidazol-2-yl)benzoic acid
3-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]-2,1-benzoxazole
1-{7-methylthieno[3,2-d]pyrimidin-4-yl}-N-[1-(pyrazin-2-yl)propan-2-yl]piperidin-4-amine
2-{[4-(2-amino-6-methylpyrimidin-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
1'-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
1-[1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
3-(3-{[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-1H-indol-1-yl)propanamide
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-4-(1H-imidazol-1-yl)benzamide
N-(adamantan-2-yl)-1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
6-ethyl-2-oxo-N-[(3,4,5-trimethoxyphenyl)methyl]-1,2-dihydropyridine-4-carboxamide
[2-(3-methoxyphenoxy)ethyl](methyl)[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amine
8-fluoro-2-({[2-(1,3-thiazol-2-yl)ethyl]amino}methyl)quinolin-4-ol
2-amino-4-(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)-6-(propan-2-yl)pyridine-3-carbonitrile
6-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-7-methyl-4-(3-methylphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
N,N-dimethyl-3-[4-(1H-pyrazol-1-yl)phenyl]-1H-1,2,4-triazol-5-amine
4-(7-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
4-({1-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]pyrrolidin-3-yl}methyl)benzoic acid
ethyl 4-[4-(5-benzamido-1H-pyrazol-1-yl)piperidin-1-yl]piperidine-1-carboxylate
10-methoxy-5-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
(1S,5R)-3-(2-fluorobenzenesulfonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[4-(methylsulfanyl)phenyl]-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(1-{4-[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,3-triazol-4-yl]phenyl}ethyl)dimethylamine
N3-cyclohexyl-1-cyclopropyl-4-oxo-N5-[(4-phenyloxan-4-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-(3-phenylpropyl)-5-(pyrimidine-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(2S,4S)-4-amino-N,N-diethyl-1-(3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carbonyl)pyrrolidine-2-carboxamide
2-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1H-1,3-benzodiazole-4-carboxamide
(1S,6R)-9-(5-methyl-4-phenylthiophene-3-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
5,6-dimethyl-3-[4-(oxolan-2-ylmethyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
(2S)-1-({4-[6-(dimethylamino)pyridazin-3-yl]phenyl}methyl)pyrrolidine-2-carboxylic acid
4-[(dimethylamino)methyl]-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]azepan-4-ol
methyl 3-benzamido-5-{[(2E)-2-methylbut-2-en-1-yl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1-methylpiperidine-2-carboxamide
1-(2-methoxy-4-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
4-[(4-methyl-5-{1-[3-(methylsulfanyl)propyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
(4aS,8aR)-6-(6-aminopyridine-3-carbonyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one