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3-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-1-ethyl-6-methyl-1,2-dihydropyridin-2-one
[1-(1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)piperidin-4-yl]methanol
N-[3-(4-fluorophenyl)propyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[2-(4-fluorophenyl)ethyl]acetamide
(2R)-2-amino-N-[2-(7-methyl-1H-indol-3-yl)ethyl]-2-phenylacetamide
4-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-N,N-dimethylaniline
(1S,6R)-9-(pyrimidin-5-ylmethyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propan-1-one
3-[(3S,4R)-1-benzyl-4-(4-methylpiperazin-1-yl)piperidin-3-yl]-N-[3-(dimethylamino)phenyl]propanamide
1,5-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-indole-2-carboxamide
8-fluoro-N-(3-hydroxy-1-phenylpropyl)quinoline-2-carboxamide
3-(3-fluorophenyl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]propan-1-one
4-{4-[(1H-indol-2-ylmethyl)amino]piperidin-1-yl}-N-(pyridin-3-ylmethyl)benzamide
N-[1-(1-cyclohexylpiperidin-4-yl)-1H-pyrazol-5-yl]-2,2-dimethylpropanamide
3-(2,5-difluorobenzoyl)-1-(dimethyl-1,3-thiazole-5-carbonyl)piperidine
[(3R,4R)-1-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
3-[1-(3,5-dimethyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridine-3-carboxylic acid
5-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}pyrazin-2-ol
7-(2-methoxyethyl)-2-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-{1-[1-(1-acetylpiperidin-4-yl)piperidin-4-yl]-2-(2-fluorophenyl)ethyl}-N-methylthiophene-3-carboxamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-3-(2-methyl-1,3-thiazol-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
3-benzyl-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperazin-2-one
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-cyclobutylpropanamide
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
methyl (1S,3S,3aR,6aS)-3-(2-hydroxy-5-methylphenyl)-5-methyl-4,6-dioxo-1-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-amino-N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-2-methylpropanamide
2-{[4-(benzyloxy)piperidin-1-yl]methyl}pyridine
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-3,3-dimethylcyclohexan-1-amine
N2-[2-(4-methylphenyl)propan-2-yl]pyrrolidine-1,2-dicarboxamide
3-[(2R,3R,6R)-5-[5-(methoxymethyl)furan-2-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
5-{3-[3-(3-methylbutyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]-3-oxopropyl}imidazolidine-2,4-dione
1-[1-(2-fluoro-4-methylbenzoyl)piperidin-4-yl]-3-phenylpropan-1-ol
3-benzyl-N-[2-(furan-2-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-(4-{1-[2-(dimethylsulfamoyl)ethyl]-1H-imidazol-2-yl}phenyl)acetamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)propanamide
3-phenoxy-N-[1-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]propanamide
2-(propan-2-yl)-4-{1-[1-(thiophen-2-yl)ethyl]-1H-imidazol-2-yl}-1,3-oxazole
1-(pyridin-3-ylmethyl)-4-[3-(pyridin-4-yl)azetidine-1-carbonyl]pyrrolidin-2-one
3-[2-({[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]carbamoyl}amino)phenyl]-N,N-dimethylpropanamide
4-{[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]amino}-2-methoxypyridine-3-carbonitrile
4-(4-ethoxyphenyl)-2-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1H-imidazole
6-[3-(7-cyclobutanecarbonyl-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
2-[2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
8-(1-benzofuran-2-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 4-(5-{[(2-hydroxyethyl)(thiophen-2-ylmethyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2,7,8-trimethylquinoline-4-carboxamide
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]cyclohexanecarboxamide
3-methyl-N-{2-[2-(quinolin-4-yl)-1H-imidazol-1-yl]ethyl}pyridin-4-amine
N-(1-{7-[(2-chloro-6-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxypropanamide