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3-({[4-(3-hydroxy-3-methylbutyl)phenyl]formamido}methyl)-1,2,4-oxadiazole-5-carboxamide
N-cyclopropyl-2-ethyl-7-(4-methylpiperazine-1-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(3-chloro-4-methoxyphenyl)-3-[(1R,2S)-2-(methoxymethyl)cyclopentyl]urea
5-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]-N-methyl-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-{4-[(2-fluorophenyl)methyl]morpholin-3-yl}-1-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
N-cyclopropyl-5-{pyrazolo[1,5-a]pyridine-3-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(3S,4R)-4-methyl-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidine-3,4-diol
1-{3-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propyl}-1H-pyrazole
6-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}pyridine-3-carboxamide
N-cyclopentyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(4aS,8aS)-2-[(4-methyl-1H-imidazol-2-yl)methyl]-decahydroisoquinolin-4a-ol
N-({1-[2-(pyrrolidin-1-yl)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-hydroxyethan-1-one
8-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[cyclopropyl(pyridin-2-yl)methyl]-N,2,7,8-tetramethylquinoline-4-carboxamide
8-chloro-2-{[4-(pyridin-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}quinoline
4-{[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]amino}-N-(propan-2-yl)pyridine-2-carboxamide
1-[2-methoxy-4-({methyl[(2-methylpyridin-4-yl)methyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
2-[2-(2-methoxyethyl)piperidine-1-carbonyl]-3,5,7-trimethyl-1H-indole
5-{4-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}quinoxaline
2-(3-fluoro-4-hydroxyphenyl)-1-[2-(3-methoxypropyl)piperidin-1-yl]ethan-1-one
N-[(5-methylpyrazin-2-yl)methyl]-2,3-dihydro-1H-indene-1-carboxamide
methyl 6-(cyclopent-1-ene-1-carbonyl)-2-[(2-phenylethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-[(5-{[benzyl(methyl)amino]methyl}-1,2-oxazol-3-yl)formamido]-N,2-dimethylpropanamide
3-[4-(pyridin-4-yl)piperidin-1-yl]-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazine
4-[1-(3-methoxybenzoyl)piperidine-4-carbonyl]-1-methylpiperazine-2-carboxylic acid
2-cyclopentyl-9-[6-(1-hydroxyethyl)pyridin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
N2-[2-(phenylsulfanyl)ethyl]-N2-(propan-2-yl)pyrrolidine-1,2-dicarboxamide
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(1H-1,3-benzodiazol-1-yl)-1-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}ethan-1-one
N-[(2-hydroxyadamantan-2-yl)methyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
9-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(2-{[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]methyl}quinolin-5-yl)acetamide
(5S,9aS,9bS)-2-(3-methoxyphenyl)-5-(4-methylphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-{2-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]ethyl}pyrrolidin-2-one
4-(4-{[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]amino}piperidin-1-yl)-N,N-dimethylbenzamide
3-[(oxolan-3-ylmethyl)sulfamoyl]-N-(2,2,2-trifluoroethyl)benzamide
N-[1-(1-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-3-methylbutanamide
2-{1-[(1-methyl-1H-imidazol-5-yl)methyl]azetidin-3-yl}-1H-1,3-benzodiazole
2-(4-acetylphenoxy)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
1-(2-ethoxyethyl)-3-methyl-N-[1-(pyridin-2-ylmethyl)azepan-3-yl]-1H-pyrazole-5-carboxamide
5-{2-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
1-(2-{[(5-tert-butyl-1H-pyrazol-3-yl)methyl]amino}pyrimidin-4-yl)pyrrolidin-3-ol
3-({cyclopropyl[(4-ethoxyphenyl)methyl]amino}methyl)-N-methylpyridin-2-amine
6-methyl-1-(oxolan-2-ylmethyl)-2-(2-phenylethyl)-3-(piperidine-1-carbonyl)-1,4-dihydropyridin-4-one
2-(4-methylpyrimidin-2-yl)benzonitrile
methyl 4-[({1-[3-(pyridine-4-amido)phenyl]piperidin-4-yl}amino)methyl]benzoate
2-amino-6-(oxolane-2-carbonyl)-4-(thiophen-3-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
8-(4,6-dihydroxypyridine-3-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one