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4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidine
6-{[benzyl(methyl)amino]methyl}-2-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-dihydropyridine-3-carboxamide
2-({cyclopropyl[(2-methoxyphenyl)methyl]amino}methyl)-4-hydroxyquinoline-6-carboxamide
6,6-dimethyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-5-oxothiomorpholine-3-carboxamide
5-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylic acid
2-[4-(2,1,3-benzothiadiazol-5-ylmethyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
(1S,5R)-3-(4,6-dimethoxypyrimidin-2-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4,6-dimethyl-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[2-(2,2-diphenylethyl)morpholin-4-yl]-3-(1H-pyrazol-4-yl)propan-1-one
7-methyl-3-(pyrimidin-4-yl)-1H-indole
3-(5-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
N-{1-[(4,8-dimethoxynaphthalen-1-yl)methyl]pyrrolidin-3-yl}acetamide
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
N-(oxolan-2-ylmethyl)-7-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N4-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-N2,N2-dimethyl-5,6,7,8-tetrahydroquinazoline-2,4-diamine
7,7-dimethyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
1-(3-chlorophenyl)-4-[2-(3-fluorophenoxy)acetyl]piperazin-2-one
4-{[3-(2,2-dimethylpyrrolidine-1-carbonyl)-1,2-oxazol-5-yl]methyl}morpholine
1-[3-(4-chlorophenyl)-3-phenylpropanoyl]piperidine-4-carboxamide
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4-(3-methylpyridin-4-yl)-1,4-diazepane
N-(cyclohex-1-en-1-ylmethyl)-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
N-{3-hydroxy-1-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-1-oxopropan-2-yl}acetamide
2-[(1S,5R)-3-(4-aminopyrimidin-2-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
2-(5-cyclohexyl-1H-1,2,4-triazol-3-yl)-N,N-bis(propan-2-yl)benzamide
2-{4-[2-(5-acetylthiophen-3-yl)acetyl]morpholin-3-yl}acetic acid
(2R)-2-({3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]phenyl}formamido)propanamide
ethyl 2-({2-[4-(4-methylphenyl)piperazine-1-carbonyl]phenyl}amino)acetate
6-(3-methyl-1H-pyrazol-1-yl)-2H-1,3-benzodioxole-5-carboxamide
5-(2-oxo-2-{4-[(prop-2-en-1-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{7-[(2,3-dimethoxyphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}propane-1,2-dione
N-methyl-N-{[3-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}cyclopropanesulfonamide
4-{3-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}phenol
{4-[4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-2-yl]-1,4-oxazepan-6-yl}methanol
N-[1-(2-chlorophenyl)cyclopropyl]-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[(2-hydroxyethyl)[(4-{[(4-methylphenyl)methyl]amino}quinazolin-2-yl)methyl]amino]ethan-1-ol
(2R,3R,6R)-5-[(2-ethylpyrimidin-5-yl)methyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(dimethylamino)-N-(2-hydroxyethyl)-2-(2-methylphenyl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
(3S,4S)-1-(4-methoxybenzoyl)-4-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]pyrrolidin-3-ol
1-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-3-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-6-yl}urea
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]({2-[2-(4-methylpiperazin-1-yl)ethoxy]phenyl}methyl)amine
2,6-dimethoxy-N-({5-methyl-2-[3-(propane-2-sulfonamido)phenyl]-1,3-oxazol-4-yl}methyl)pyridine-3-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(2-methyl-5-sulfamoylphenyl)pyrrolidine-1-carboxamide
[(3R,4R)-1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
5-[2-(azepan-1-yl)acetyl]-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-ethyl-2,3-dimethyl-N-[(5-methylpyrazin-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-[4-(1,3-benzothiazol-2-yl)-1,4-diazepan-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
N-(2-methylpropyl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-(thiophen-3-ylmethyl)propanamide
2-methoxy-6-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}phenol
N-cyclopentyl-2-{[(2,3-difluoro-4-methoxyphenyl)methyl]amino}propanamide