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1-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclopentan-1-ol
4-{[methyl({[2-(trifluoromethyl)phenyl]methyl})amino]methyl}benzene-1,2-diol
2-(2-chloro-4-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}phenoxy)acetamide
6-chloro-2-{[3-(pyrrolidin-1-yl)piperidin-1-yl]methyl}quinoline
1-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-4-(1H-1,2,3,4-tetrazol-5-yl)piperidine
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-({[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]amino}methyl)piperidin-2-one
2-ethyl-6-methyl-3-{[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methoxy}pyridine
2-methyl-6-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridine
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-6-methyl-4-oxo-N-(oxolan-2-ylmethyl)-4H-pyran-2-carboxamide
5-(1H-1,3-benzodiazol-1-yl)pyrazin-2-amine
1-{1-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]piperidin-4-yl}-3-methylbutan-1-ol
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-{[2-(propylamino)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]methanol
2-{5-[5-(1H-1,3-benzodiazol-1-ylmethyl)-1H-pyrazole-3-carbonyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
6-{[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]methyl}naphthalen-2-ol
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]but-2-ynamide
({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)(pyridin-3-ylmethyl)amine
5-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
5-[4-(4-acetylphenyl)piperazin-1-yl]-1-ethyl-N-(furan-3-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[(1R)-1-phenylethyl]urea
4-[(1-acetylpiperidin-4-yl)oxy]-N-[(5-ethylpyridin-2-yl)methyl]-3-methoxybenzamide
2-[(2-chlorophenyl)methyl]-4-(3-propyl-1H-pyrazole-4-carbonyl)morpholine
[(3R,4R)-4-[(dimethylamino)methyl]-1-[4-(2-methylphenyl)benzoyl]pyrrolidin-3-yl]methanol
methyl 4-{4-[(4-cyclohexyl-3-oxopiperazin-1-yl)methyl]-5-methyl-1,3-oxazol-2-yl}benzoate
2,6-dimethyl-5-{2-oxo-2-[3-(pyridin-4-yl)azetidin-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methoxy-2-methylbenzamide
4-methyl-2-{1-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]piperidin-4-yl}-1H-1,3-benzodiazole
ethyl(oxolan-2-ylmethyl){[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
2-(1H-indole-5-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
[(3R,4R)-1-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine
(1R,3S)-7-(2,5-dimethyl-1-phenyl-1H-pyrrole-3-carbonyl)-3-ethoxy-7-azaspiro[3.5]nonan-1-ol
N-(1-{5-[(cyclohexylmethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)cyclobutanecarboxamide
N,2-dimethyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
2-[5-(3-methylthiophen-2-yl)-4-phenyl-1H-imidazol-1-yl]-1-(pyridin-3-yl)ethan-1-ol
N,N-dimethyl-3-{[3-(1H-1,2,3-triazol-1-yl)propyl]sulfamoyl}benzamide
(2R,6R)-4-(3-methoxypropanoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-3-(3,5-dimethylphenyl)propanamide
3-methoxy-1-[3-(4-phenoxybenzoyl)piperidin-1-yl]propan-1-one
2-butyl-N-methyl-N-[2-(morpholin-4-yl)ethyl]-1,3-benzoxazole-5-carboxamide
methyl({[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-(pyrrolidin-1-ylmethyl)-1-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidine
4-chloro-N,N-dimethyl-5-{1-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-imidazol-2-yl}-1,3-thiazol-2-amine
2-[2-(trifluoromethyl)morpholin-4-yl]-1,3-thiazole-4-carboxamide
N-[(3R,4S)-1-[(4,4-dimethylpiperidin-1-yl)sulfonyl]-4-propylpyrrolidin-3-yl]acetamide
8-(3-methylquinolin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
2-(2,5-dimethoxyphenyl)-5-methyl-4-{1H-pyrazolo[3,4-b]pyridin-1-ylmethyl}-1,3-oxazole
[(3R,4R)-1-benzoyl-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-2-(5-fluoro-2-methyl-1H-indol-3-yl)acetamide
N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)quinoline-2-carboxamide