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N,N-dimethyl-7-(3-methyl-1H-pyrazole-5-carbonyl)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[3-(1H-pyrazol-1-yl)benzoyl]-4-[2-(pyridin-2-yl)ethyl]piperazine
2-({[(3R,4R)-4-(hydroxymethyl)-1-(quinolin-6-ylmethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl](methyl)[1-(pyridin-3-yl)propyl]amine
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[2-(1H-pyrrol-1-yl)ethyl]piperazine
2-{[(1-hydroxybutan-2-yl)(thiophen-3-ylmethyl)amino]methyl}benzonitrile
6-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-N-[(4-phenyloxan-4-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
(4aR,8aR)-2-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
2-methyl-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-2-(1H-pyrrol-1-yl)propanamide
2-ethyl-8-({1-methyl-4-oxo-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-6-yl}methyl)-2,8-diazaspiro[4.5]decan-3-one
methyl 2-(4-{[1-(methylsulfanyl)propan-2-yl]amino}piperidin-1-yl)acetate
1-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-3-[3-(1H-1,2,4-triazol-1-yl)propyl]urea
N-(5-methyl-2-pentanamidophenyl)-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-cyclopropyl-N-({3-[(1-methylpiperidin-3-yl)methoxy]phenyl}methyl)thiophene-2-carboxamide
1-[(2-fluorophenyl)methyl]-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-6-oxopiperidine-3-carboxamide
5-(cyclopropylamino)-1-methyl-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-ethyl-2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
N,N-dimethyl-1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]pyrrolidin-3-amine
1-[(3-methyl-1,2-oxazol-5-yl)methyl]-8-(2-methylquinolin-4-yl)-1,8-diazaspiro[4.5]decane
1-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]-2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}ethan-1-one
3,5-dimethyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1-benzofuran-2-carboxamide
5-(4-chloro-2-methoxyphenoxymethyl)-N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
3-(5-{1-[3-(1,3-thiazol-4-yl)phenyl]-1H-imidazol-2-yl}thiophen-2-yl)prop-2-yn-1-ol
2-{4-[(3-methyl-1H-pyrazol-5-yl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
1-[1-(3,5-dimethylfuran-2-carbonyl)piperidin-3-yl]-4-(4-fluorophenyl)piperazine
N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-3-methyl-5,6-dihydro-1,4-dioxine-2-carboxamide
(2S)-2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)-3-phenylpropanamide
(1-{4-[4-({[4-(trifluoromethoxy)phenyl]methyl}amino)piperidin-1-yl]benzoyl}piperidin-3-yl)methanol
2-[(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]-5-methoxy-4H-pyran-4-one
(1R,5R)-6-(cyclobutylmethyl)-3-(2-methylpyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonane
(3S,4R)-1-[2-(3-fluorophenoxy)acetyl]-4-phenylpyrrolidine-3-carboxylic acid
N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
[4-(quinoxalin-2-yl)-1,4-oxazepan-6-yl]methanol
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)cyclobutanecarboxamide
N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-3-(4-methylphenyl)-1H-pyrazole-5-carboxamide
(1S,5R)-6-[(4-chloro-3-fluorophenyl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-(propan-2-yl)pyrimidine
N-(2,3-dihydro-1-benzofuran-5-ylmethyl)-4-methyl-5-(1-methyl-1H-pyrazol-3-yl)-1,3-thiazol-2-amine
4-(dimethyl-1,2-oxazol-4-yl)-3-[2-(phenylamino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(4-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)-2,5-dimethylpyrazine
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(4-phenylbenzoyl)piperidine
(3R,4R)-1-(2-methoxyquinoline-4-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
ethyl 4-{[3-(4-tert-butylbenzoyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
N-(2-{7-[(2-chloro-6-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methoxybenzamide
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-(2-cyclopropylpyrimidin-5-yl)-N,N,7,8-tetramethylquinoline-4-carboxamide
4-ethyl-1-(3-phenylpropyl)-1,4-diazepan-5-one
methyl 5-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-5-oxopentanoate
3-[5-chloro-2-(1H-1,2,4-triazol-1-yl)phenyl]-1-{[4-(dimethylamino)oxan-4-yl]methyl}urea