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N-ethyl-3-(pyridin-2-yl)-3-(pyridin-4-yl)propanamide
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
7-(6-oxo-1-propylpiperidine-3-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
3-(3-methoxyphenyl)-1-[2-(2-phenylethyl)morpholin-4-yl]propan-1-one
(4S)-4-acetamido-4-[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]butanamide
4-(cyclopropylmethyl)-1-(3-methylfuran-2-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-(pyridazine-3-carbonyl)piperidin-4-ol
1-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
1,5-dimethyl-N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1H-pyrazole-3-carboxamide
N-(1-hydroxypropan-2-yl)-4-{[2-(2-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
4-methyl-5-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,3-oxazole
1-{2-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-oxoethyl}-3-methyl-1,2-dihydroquinoxalin-2-one
methyl 2-[(2-methylpropyl)sulfamoyl]-6-[3-(prop-2-en-1-yloxy)benzoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(3S,4R)-1-({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)-3-methoxypiperidin-4-amine
1-methyl-4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperazine-2-carboxylic acid
2-ethyl-3-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6-methyl-1-[(5-methylfuran-2-yl)methyl]-1,4-dihydropyridin-4-one
9-[2-(benzyloxy)acetyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-2-[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]pyridine-4-carboxamide
4-{4-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}amino)methyl]phenyl}but-3-yn-1-ol
5-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidine-1-carbonyl]pyridine-2-carbonitrile
2-(pyridin-4-yl)-7-(quinoline-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-[2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)ethyl]benzene-1-sulfonamide
1-methyl-2-(1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}piperidin-3-yl)-1H-1,3-benzodiazole
N-[(1-cyclopentylpiperidin-3-yl)methyl]-1-ethyl-3-methyl-N-[2-(piperidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
(2S,4R)-4-(4-{[1-(3-fluorophenyl)-N-methylformamido]methyl}-1H-1,2,3-triazol-1-yl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-5-methyl-2-oxopiperazin-1-yl]benzonitrile
5-(2-fluorophenyl)-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-1,2,4-triazin-3-amine
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-(furan-2-yl)-2-oxoacetamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(propane-1-sulfonyl)-2,8-diazaspiro[4.5]decan-3-one
ethyl 1-{2-[(4-methylpyridin-2-yl)amino]ethyl}-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
2-phenyl-2-{2-[1-(propan-2-yl)piperidin-4-yl]acetamido}acetic acid
methyl 3-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-1-(2-methoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
4-methylphenyl (7S,9aR)-7-[(1R)-1-hydroxyethyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}acetamide
N-[1-(3-phenylpropyl)piperidin-3-yl]-3-(pyrazin-2-yl)propanamide
2-{[(1R,5S,8S)-8-hydroxy-3-azabicyclo[3.2.1]octan-3-yl]methyl}-5,8-dimethylquinolin-4-ol
N-[(2-aminopyridin-3-yl)methyl]-4-(piperidin-3-yl)benzamide
N-[(3S,7S,8aS)-3-(cyclohexylmethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methoxybenzamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
methyl 1-(2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetyl)piperidine-4-carboxylate
N-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-1-(thian-4-yl)piperidin-4-amine
2-(5-amino-1,3,4-thiadiazol-2-yl)-N-[(2-chlorophenyl)methyl]-N-(prop-2-en-1-yl)acetamide
5-(6-chloro-2H-chromen-3-yl)-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
5-(2,6-dimethoxyphenyl)-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1,2,4-triazin-3-amine
(4aR,8aR)-2-cyclopentanecarbonyl-7-(4-methylphthalazin-1-yl)-decahydro-2,7-naphthyridin-4a-ol
3-({2-[1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
(3R,4R)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3,4-dimethylpyrrolidin-3-ol
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-2-{3-oxo-2-azaspiro[4.4]nonan-2-yl}acetamide
3-methoxy-N-[2-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)ethyl]benzamide
2-(dimethyl-1,3-thiazol-4-yl)-1-(4-{[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)ethan-1-one