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3-acetamido-N-[1-(3-phenylpropyl)piperidin-3-yl]benzamide
2-(2-hydroxyethyl)-9-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{1-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]azetidin-3-yl}morpholine
5-(3,3-diphenylpiperidine-1-carbonyl)-2-methylpyrimidine
N3-(cyclohexylmethyl)-4-oxo-1-(propan-2-yl)-N5-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-{1-[1-(3-cyclohexylpropanoyl)piperidin-4-yl]-2-phenylethyl}-N-cyclopropylpyridine-2-carboxamide
1-{2-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}azepan-2-one
N-cyclopropyl-1-{1-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]piperidin-4-yl}piperidine-3-carboxamide
6-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-N-[2-(4-methoxyphenyl)ethyl]-5-methylthieno[2,3-d]pyrimidin-4-amine
1-(4-{[3-(pentan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenyl)-1H-1,2,4-triazole
1-(9H-purin-6-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]piperidin-4-amine
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]propan-1-one
1-[4-({[3-(1H-indazol-1-yl)propyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
N-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,3-difluorobenzamide
(3S,4S)-4-methyl-1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidine-3,4-diol
N-methyl-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}-N-[2-(pyrrolidin-1-yl)ethyl]acetamide
2-{1-[2-(4-fluorophenoxy)ethyl]pyrrolidin-3-yl}benzoic acid
2-[2-(4-fluorophenoxymethyl)pyrimidin-4-yl]pyridine-4-carboxylic acid
4-{[(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)amino]methyl}-6-ethyl-2H-chromen-2-one
2-[4-(acetamidomethyl)piperidin-1-yl]-2-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}acetic acid
1-(2-phenylethyl)-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-(oxan-4-yl)piperazin-2-yl}ethan-1-ol
1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
2-(2-aminoethyl)-N-benzyl-N-methylquinazolin-4-amine
2-{5-[1-(ethylsulfanyl)ethyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
3-{2-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
N-[2-(1-benzylpyrrolidin-3-yl)ethyl]-4-hydroxy-1-methylpiperidine-4-carboxamide
4-(1-{1-[(2-methylphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
5-(1-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-imidazol-2-yl)-2-(pyrrolidin-1-yl)pyrimidine
6-[2-(2,2-diphenylethyl)morpholine-4-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
N,N-dimethyl-2-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-2,3-dihydro-1H-inden-2-amine
methyl[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(3-hydroxy-2,2-dimethylpropyl)piperidine-3-carboxamide
methyl({[5-(1H-pyrazol-3-yl)furan-2-yl]methyl})(thiophen-3-ylmethyl)amine
2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[2-(5-methylfuran-2-yl)ethyl]acetamide
3-[5-(1-methyl-1H-pyrazol-4-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-[3-(cyclohexylsulfanyl)propyl]-2-(dimethyl-1,3-thiazol-5-yl)acetamide
2-(1-{[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
1-{1'-[4-(hydroxymethyl)benzoyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
4-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}benzonitrile
5-[3-(diethylamino)pyrrolidine-1-carbonyl]-N-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
3-benzyl-5-{[2-(ethylsulfanyl)-1,3-thiazol-4-yl]methyl}-1H-1,2,4-triazole
1-(cyclohex-3-en-1-ylmethyl)-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
5-fluoro-2-[5-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]-3-methyl-1H-indole
6-(2,6-dimethoxyphenyl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
methyl 1-benzyl-5-[(5-methylhex-5-en-2-yl)amino]-3-(oxolane-2-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-[3-(hydroxymethyl)piperidine-1-carbonyl]-5-methoxybenzoic acid
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(6-methylpyridazin-3-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,2,6-trimethylpyrimidine-4-carboxamide