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(2S)-2-amino-1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-4-(methylsulfanyl)butan-1-one
(1S,5R)-3-(pyridin-3-ylmethyl)-6-{[3-(trifluoromethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N,3,6,7-tetramethyl-N-[2-(oxan-2-yl)ethyl]-1-benzofuran-2-carboxamide
N-[1-(pyridin-2-yl)propan-2-yl]-2-(pyridin-4-yl)quinoline-4-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamide
7-{[3-(3,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-oxa-7-azaspiro[4.5]decane
4-(1-benzyl-1H-imidazol-2-yl)-1-(2-methyloxane-2-carbonyl)piperidine
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-1,2-oxazole-3-carboxamide
3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(propane-1-sulfonyl)piperidine
4-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1-methylpiperidin-4-ol
9-(2-hydroxy-4-methylpentanoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(2-methoxyethyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
(1r,4r)-4-[2-(2,4,5-trimethoxyphenyl)-1H-imidazol-1-yl]cyclohexan-1-ol
N-[2-(dimethylsulfamoyl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
4-[1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine-4-carbonyl]morpholine
2,3-dimethyl-6-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
5-[(2-fluorophenyl)methyl]-5-(piperidin-4-yl)-3-(pyrazin-2-ylmethyl)imidazolidine-2,4-dione
N-cyclobutyl-2-(4-methylpyridine-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
5-{[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]methyl}-N-methylfuran-2-carboxamide
2-ethoxy-5-(2-{[(5-methylpyrazin-2-yl)methyl]amino}pyrimidin-4-yl)benzoic acid
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-(4-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
1-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-4-(morpholin-4-yl)butan-1-one
9-(2-hydroxy-5-methylbenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(2-chloro-4-fluorobenzoyl)-1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[3-(methylsulfanyl)propyl]propanamide
4-hydroxy-N,2-dimethyl-N-[(4-phenylphenyl)methyl]pyrimidine-5-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(pyridin-2-ylmethyl)piperidin-3-amine
2-methoxy-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyridine-4-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
N-{2-[(2-chlorophenyl)formamido]ethyl}-2-(1H-imidazol-2-yl)benzamide
N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-2-(trifluoromethyl)pyrimidin-4-amine
(1S,6R)-9-[2-(4-methanesulfonylphenyl)acetyl]-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
4-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
4-cyano-1-methyl-N-(piperidin-3-ylmethyl)-1H-pyrrole-2-carboxamide
3,5,7-trimethyl-2-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]-1H-indole
8-benzyl-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-methoxy-1-[(3-propyl-1H-pyrazol-5-yl)methyl]piperidine
(2S)-4-methyl-2-phenyl-1-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}piperazine
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}-3-(morpholin-4-yl)propan-1-one
ethyl 1-(4-methylbenzenesulfonyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
1-[(3-methoxyphenyl)methyl]-4-[5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperazin-2-one
N,N-dimethyl-6-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyrazine-2-carboxamide
N-[(3-hydroxypiperidin-3-yl)methyl]-3,5-bis(trifluoromethyl)benzamide
N-[(3,4-difluorophenyl)methyl]-2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
[(1-cyclohexylpiperidin-3-yl)methyl][(4-fluoro-2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
2-{[1-(dimethylamino)propan-2-yl]amino}-N-(propan-2-yl)acetamide
6-{[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-({[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)-N-methylacetamide
N-(4-fluorophenyl)-1-(1H-indazole-3-carbonyl)piperidin-3-amine