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N-[2-(2,4-dimethoxyphenyl)ethyl]-5-(3-fluoro-4-methoxyphenyl)-1,2,4-triazin-3-amine
1-[benzyl(methyl)amino]-3-[4-({[2-(diethylamino)ethyl]amino}methyl)phenoxy]propan-2-ol
(1S,5R)-6-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3R,4S)-4-cyclopropyl-1-[2-(2-oxoazepan-1-yl)acetyl]pyrrolidin-3-yl]methanesulfonamide
1-{4-[3-(2,5-dimethylfuran-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]phenyl}-1H-pyrazole
5-{[2-(1-ethyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-methoxy-N-[3-(pyridin-4-yl)phenyl]acetamide
1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-(4-fluorophenyl)piperazine
N-methyl-5-[1-(3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-1-phenylcyclohexane-1-carboxamide
N-{3-chloro-4-[(propan-2-yl)carbamoyl]phenyl}-2-ethyl-2,5-dihydro-1H-pyrrole-1-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)acetamide
1-[2-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidin-4-yl)ethyl]pyrrolidin-2-one
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]piperidin-3-yl]propan-1-ol
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-imidazol-1-yl)ethyl]methylamine
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-(thiomorpholin-4-yl)pyridine-3-carboxamide
4-{2-[4-(pyridin-4-yl)piperidine-1-carbonyl]phenyl}morpholine
3-{2-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethyl}-1H-indole
3-(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-4-yl)-1-(pyrrolidin-1-yl)propan-1-one
2-chloro-N-{1-[1-(cyclohexylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
2-[2-(3-methoxyphenyl)ethyl]-4-(4-propanoylpiperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-2,6-dimethoxybenzamide
2-ethyl-1-methyl-4-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]piperazine
3-{[3-(1H-pyrazol-1-yl)phenyl]formamido}-N-(1,3-thiazol-2-yl)propanamide
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1H-pyrazol-5-ylmethyl)amine
3-[benzyl({[2-(methylamino)pyridin-3-yl]methyl})amino]-2-methylpropan-1-ol
1-[(4aR,8aS)-6-(pyridine-2-carbonyl)-decahydro-1,6-naphthyridin-1-yl]-2-cyclopentyl-2-phenylethan-1-one
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(1-phenyl-1H-pyrazol-4-yl)methyl]amine
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(3-phenoxyphenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
5-(3-acetamidophenyl)-N-(4-methoxyphenyl)furan-2-carboxamide
({5-[1-(1,3-benzothiazol-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
methyl 4-{[4-(4-methoxybenzoyl)piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylate
(3S,4S)-4-cyclopropyl-1-[(dimethyl-1,3-thiazol-2-yl)methyl]pyrrolidine-3-carboxylic acid
5-(3-fluoro-2-methoxybenzoyl)-3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
7-{[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]methyl}-2-(methylsulfanyl)-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-5-phenyl-1,2-oxazole-3-carboxamide
N-ethyl-2-(4-fluoro-3-methylphenyl)pyridine-4-carboxamide
5-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]pyrazin-2-ol
N-{1-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-2-(2-fluorophenyl)ethyl}-N-methylthiophene-3-carboxamide
(2R,3S,6R)-3-phenyl-5-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{3-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidine-1-carbonyl]-5-methylthiophen-2-yl}-2,2-dimethylpropanamide
2-methyl-7-{[5-(1,2-oxazol-3-yl)thiophen-2-yl]sulfonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
1-(2-hydroxyethyl)-5-(1H-indol-3-ylmethyl)-N-(1-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-(4-{[1-(prop-2-en-1-yl)-1H-1,3-benzodiazol-2-yl]methyl}piperazin-1-yl)-9H-purine
4-(2-methoxyphenoxy)-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidine
N-[2-(4-fluorophenyl)-1-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}ethyl]-2-methoxy-N-methylacetamide
1-{7-methanesulfonyl-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-2,5-dihydro-1H-pyrrole
N-ethyl-2-{4-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]piperazin-1-yl}pyrimidin-4-amine