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(4S)-4-(propan-2-yl)-3-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-1,3-oxazolidin-2-one
2-(diethylamino)-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)acetamide
3-{[1-(1-benzoxepine-4-carbonyl)pyrrolidin-3-yl]methyl}benzamide
3-[4-(dimethylamino)azepane-1-carbonyl]-6-methyl-1,4-dihydroquinolin-4-one
(3S,4S)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-N-methylpyridine-3-carboxamide
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
2-oxo-N-[(1R,3S)-3-[(2,2,2-trifluoroethyl)carbamoyl]cyclopentyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-methyl-N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
2-benzyl-4-[(E)-2-phenylethenesulfonyl]morpholine
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-2-(2-methoxyphenyl)-1,3-thiazole
N-[2-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]thiomorpholine-4-carboxamide
N-(2,2-diphenylethyl)-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[(dimethylamino)methyl]-N-[(1-methylpyrrolidin-3-yl)methyl]-1,3-thiazole-4-carboxamide
2-amino-4-(2,5-dimethoxyphenyl)-7-methyl-5H,7H-thieno[3,4-b]pyridine-3-carbonitrile
(2S,4R)-1-[(4-chlorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]pyrrolidine-2-carboxamide
methyl 8-(1H-1,3-benzodiazol-2-ylmethyl)-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-(3-hydroxypropyl)-1-{1-[(2-methoxynaphthalen-1-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
N-(1,2-oxazol-3-ylmethyl)-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
1-(furan-2-ylmethyl)-1-methyl-3-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}urea
(1R,5S,6R,7S)-6-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-3-propyl-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
2-[4-methyl-6-(methylamino)pyrimidin-2-yl]-N,N-bis(propan-2-yl)benzamide
1-methyl-3-{[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}-1,2-dihydroquinolin-2-one
5-{2-[(3,4-dimethoxyphenyl)methyl]pyrimidin-4-yl}-2-ethoxybenzoic acid
ethyl 1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxylate
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-2-fluorobenzamide
2-{1-[(2-fluorophenyl)methyl]-4-(5-propylpyrimidin-4-yl)piperazin-2-yl}ethan-1-ol
1-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)urea
8-[2-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)acetyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(1,2-benzoxazol-3-yl)-1-[4-(pyridin-3-yloxy)piperidin-1-yl]ethan-1-one
1-ethyl-N-methyl-3-(2-methylpropyl)-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
2-amino-4-(1-methyl-1H-pyrazol-4-yl)-6-(3,4,5-trifluorophenyl)pyridine-3-carbonitrile
5-fluoro-2-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-3-methyl-1H-indole
2-(4-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-1-yl)-N-ethylacetamide
2-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-6-methylpyrimidine-4-carboxylic acid
(5S,9aS,9bS)-5-(2-chloro-6-fluorophenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N,N-diethylacetamide
2,5-difluoro-N-(2-propoxypropyl)benzamide
2-(4-fluorophenyl)-N-[2-(7-{[3-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]acetamide
3-fluoro-N-[2-(2-hydroxyethoxy)ethyl]-5-methylimidazo[1,2-a]pyridine-2-carboxamide
1-{[2-methoxy-4-(4-methoxy-3-methylphenoxy)phenyl]methyl}pyrrolidine
(3R,4S)-4-(4-methoxyphenyl)-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]pyrrolidin-3-amine
2-(4-chlorophenyl)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}acetamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[(6-methyl-2-propylpyrimidin-4-yl)amino]pyrrolidin-2-one
2-{3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]piperidin-1-yl}acetamide
N-[(3R,4S)-1-[4-(1H-imidazol-1-yl)butanoyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
N-{2-[7-(1-benzothiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}oxolane-2-carboxamide
N-cyclopropyl-1-{1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidin-4-yl}piperidine-3-carboxamide
N-ethyl-4-hydroxy-2-(4-methylphenyl)-N-[2-(pyrrolidin-1-yl)ethyl]pyrimidine-5-carboxamide