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6-{[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl}-2H-chromen-2-one
methyl 2-({[1-(carbamoylmethyl)-2-methyl-1H-indol-3-yl]methyl}amino)-2-(3-methylphenyl)acetate
3-[2-(azepan-1-yl)-2-oxoethyl]-4-[(3-phenoxyphenyl)methyl]piperazin-2-one
3-chloro-4-{[1-(1H-indol-3-ylmethyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
6-[1-(2,3-dihydro-1H-indene-1-carbonyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
2-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)phenol
4-(2-phenoxyethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
1-{2-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperazin-1-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(pyrimidin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[1-(1H-imidazol-2-yl)ethyl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
3-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}-1-methyl-1H-indole
(1R,7S)-3-[2-(piperidin-1-yl)ethyl]-6-(pyrrolidine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
(1S,5R)-6-methyl-3-(3-phenoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-acetyl-N-[(3S,4R)-4-ethoxyoxolan-3-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2,3,4-trimethoxybenzamide
4-{[5-(2,5-dihydro-1H-pyrrol-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-propylpiperidine
3-[2-(dimethylamino)ethyl]-1-(3-methylbutyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-3-(2-methylphenyl)piperidine
2-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-methylacetamide
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
2-cyclopentyl-9-[(2S)-2-hydroxy-2-phenylacetyl]-2,9-diazaspiro[5.5]undecan-3-one
7-(3,4-dihydro-2H-1,5-benzodioxepine-7-sulfonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-({5-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
6-methyl-2-oxo-N-(prop-2-en-1-yl)-4-(pyridin-3-yl)-N-(pyridin-4-ylmethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
4-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
N-(2-acetamidoethyl)-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-methylpyridine-4-carbonyl)piperidin-3-ol
1-{2,7-diazaspiro[4.5]decan-2-yl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
8-(1,3-benzothiazol-2-yl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-1,8-diazaspiro[4.5]decane
4-fluoro-N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}benzene-1-sulfonamide
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-5-chloro-2-methylbenzamide
N-[3-(furan-2-yl)phenyl]-1-(oxane-2-carbonyl)piperidine-4-carboxamide
3-(4-methoxypyrimidin-2-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
3-(3-methylbut-2-en-1-yl)-1-(thiophene-3-carbonyl)piperidine-3-carboxylic acid
4-methyl-2-(5-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-3-phenyl-1H-1,2,4-triazol-1-yl)pyridine
6-(2-chlorophenyl)-2-{4-[(3-hydroxyazetidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
N-cyclopropyl-N-({3-[(1-methylpiperidin-3-yl)methoxy]phenyl}methyl)pyridine-4-carboxamide
1-(2,6-difluoro-4-methoxybenzoyl)-2-(4-fluorophenyl)piperidine
(4aS,8aS)-2-{[3-(morpholin-4-yl)phenyl]methyl}-decahydro-2,7-naphthyridin-4a-ol
2-({2-[1-(1-ethyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-cyclopropyl-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(3S,4S)-1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-(propan-2-yloxy)pyrrolidin-3-ol
{3-ethyl-1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperidin-3-yl}methanol
ethyl 1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]piperidine-3-carboxylate
3-benzyl-3-{[1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]methyl}-1-methyl-2,3-dihydro-1H-indol-2-one
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1H-pyrazole-4-carboxamide
2-(dimethylamino)-N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-4-methylpyrimidine-5-carboxamide
(3S,4S)-1-{[3-(cyclopentyloxy)phenyl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-(trifluoromethyl)benzamide