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2-{[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzonitrile
1-(3-methylpyridin-2-yl)-1H-1,3-benzodiazole
5-(ethoxymethyl)-8-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methoxy}quinoline
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-{[4-(propan-2-yl)piperidin-1-yl]methyl}piperidin-2-one
4-[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,2-dimethylpiperazine
[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl](methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
1'-(2,4-difluoro-3-methoxybenzoyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
(1S,5R)-6-(cyclopropylmethyl)-3-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-amino-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)-4-[4-(pyridin-2-yl)phenyl]pyridine-3-carbonitrile
2-propyl-N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-1,3-thiazole-4-carboxamide
4-(3-{[1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]oxy}benzoyl)morpholine
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
ethyl 4-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H-pyrazole-3-carboxylate
N,2-dimethyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-6-(piperidin-4-yl)pyrimidin-4-amine
N-[(1S,2R)-2-carbamoylcyclopentyl]-4-(3-hydroxy-3-methylbutyl)benzamide
1-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
7-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
N3-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-N1-(pyridin-3-yl)propane-1,3-diamine
N-(2-hydroxypropyl)-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
(2S,4S)-4-amino-1-[3-(4-fluorophenyl)benzoyl]pyrrolidine-2-carboxylic acid
N-methyl-5-[3-(1H-pyrazol-1-yl)phenyl]thiophene-2-carboxamide
N-(3-chloro-4-methoxyphenyl)-3-[1-(oxan-4-yl)piperidin-3-yl]propanamide
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
3-chloro-N-{[5-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-2-carboxamide
7-(3,6-dimethylpyrazin-2-yl)-4-[2-(1-methylpyrrolidin-2-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-cyclohexyl-4-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(3-methyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[1-(1-{1-[(propan-2-yl)carbamoyl]ethyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopentanecarboxamide
1-[1-(adamantane-1-carbonyl)piperidin-3-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
N-{[1-(quinolin-2-ylmethyl)-1,2,3,6-tetrahydropyridin-4-yl]methyl}acetamide
(1S,5R)-6-(3-fluoro-4-methoxybenzoyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(2S)-3-methyl-2-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}butanamide
N-[(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)methyl]acetamide
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide
1-(3-{[(7-chloroquinolin-4-yl)amino]methyl}pyridin-2-yl)piperidin-3-ol
ethyl 3-{[5-(2,6-dimethylphenoxymethyl)-1,2-oxazol-3-yl]formamido}hexanoate
2-(5-{[3-(thiophene-2-carbonyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyrazine
2-[1-(4,6-dimethylpyrimidin-2-yl)pyrrolidin-3-yl]benzoic acid
4-(4-chlorophenyl)-N-methyl-N-[2-(methylcarbamoyl)ethyl]butanamide
methyl[1-(pyridin-2-yl)ethyl]{[4-(pyridin-2-yl)phenyl]methyl}amine
5-[3,5-dimethyl-1-(1H-1,2,3,4-tetrazol-5-yl)-1H-pyrazol-4-yl]-8-methoxy-2-methylquinoline
1-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)-5-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-{5-[(2-chloro-4-fluorophenyl)methyl]-1,2,4-oxadiazol-3-yl}-6-methylpyridazine
4-[2-(4-fluorophenoxy)ethyl]-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-5-one
[(3R,4S)-1-[(2-ethylphenyl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
(5-{1-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1H-imidazol-2-yl}-2-ethoxyphenyl)methanol
1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}-3-(1,2-oxazinan-2-yl)propan-1-one
N-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
6-(4,4-dimethylpiperidin-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
4-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-2-(trifluoromethyl)morpholine