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N,N-dimethyl-3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-[(3R,4S)-3-cyclobutaneamido-4-(propan-2-yl)pyrrolidin-1-yl]propanoic acid
2-(4-fluorophenyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-(quinolin-5-ylmethyl)acetamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]propanamide
butyl 4-acetyl-4-phenylpiperidine-1-carboxylate
2-(1-methyl-4-{[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}piperazin-2-yl)ethan-1-ol
N4-(cyclohex-1-en-1-ylmethyl)-6-(4-methylpiperazin-1-yl)pyrimidine-2,4-diamine
1-[1-(4-ethenylbenzoyl)piperidin-4-yl]piperidin-3-ol
(4aS,7aR)-1-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-2-(methylsulfanyl)-N-(oxolan-2-ylmethyl)acetamide
N,2-diethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-4-methyl-1,3-oxazole-5-carboxamide
2-(4-hydroxyphenyl)-1-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethan-1-one
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-3-(1H-pyrazol-4-yl)benzamide
N-[3-(1H-imidazol-1-yl)butyl]-6-(propan-2-yl)pyrimidin-4-amine
2-(1-propylpiperidin-4-yl)-1-(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)ethan-1-one
1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(thiophen-3-yl)ethan-1-one
{4-[(4-chlorophenyl)methyl]piperidin-4-yl}methanol
6-chloro-2-(1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
(3S,4S)-4-[4-(pyridin-2-yl)piperazin-1-yl]-1-(1,3-thiazol-2-ylmethyl)pyrrolidin-3-ol
7-[(2-fluorophenyl)methyl]-2-[(5-methylfuran-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(1R,3S,5S)-8-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
3-[(2R,3R,6R)-5-(3,4-difluorobenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[(3-methoxyphenyl)methyl]-3-(1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-3-yl)propanamide
5-chloro-4-[({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]-2-methoxyphenol
5-acetyl-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)thiophene-3-carboxamide
2,6-dihydroxy-N-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]benzamide
N-[2-fluoro-5-({[3-(methylsulfanyl)propyl]carbamoyl}amino)phenyl]-2-methylpropanamide
N,N,4-trimethyl-5-[4-(4-methylphenoxy)piperidine-1-carbonyl]pyrimidin-2-amine
(3aR,7aS)-2-(4-methoxypyrimidin-2-yl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
(2S,4S)-4-amino-1-[2-(benzyloxy)acetyl]-N-ethylpyrrolidine-2-carboxamide
(3aR,6aR)-2-[2-(4-fluorophenyl)acetyl]-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[5-(2,6-dimethylpyrimidin-4-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carboxamide
N-ethyl-3-(4-methyl-1,3-thiazol-5-yl)-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)propanamide
N-{[3-(methylsulfanyl)phenyl]methyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-ethyl-3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]benzamide
(3S,4R)-1-(isoquinoline-3-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
2-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
4-(1,3-dimethyl-1H-pyrazol-4-yl)-2-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}pyrimidine
(3S,4R)-4-(4-fluorophenyl)-1-(3-methoxypropanoyl)pyrrolidine-3-carboxylic acid
3-{4-[2-(4-methanesulfonylphenyl)-1H-imidazol-1-yl]phenyl}-5-methyl-4H-1,2,4-triazole
N-[(3S,4R)-1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
N-[5-(dimethylamino)-2-methylphenyl]-2-(piperidin-1-ylmethyl)-1,4-oxazepane-4-carboxamide
2-(9-{[2-(methylsulfanyl)phenyl]methyl}-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl)acetic acid
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(pyridin-4-yl)ethyl]amine
2-[2-({7-methyl-12-oxo-3,7,11-triazaspiro[5.6]dodecan-3-yl}methyl)phenoxy]acetic acid
4-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2-(trifluoromethyl)morpholine
2-[1-(cyclohexylmethyl)-4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperazin-2-yl]ethan-1-ol
1-(2-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}ethyl)-4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperazine