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2-[1-(2-fluorophenyl)-5-(2H-1,2,3-triazol-2-ylmethyl)-1H-1,2,4-triazol-3-yl]acetamide
3-[(3S,4R)-1-benzyl-4-(4-methylpiperazin-1-yl)piperidin-3-yl]-N-[2-(dimethylamino)ethyl]propanamide
14-(1H-indol-5-yl)-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
2-(6-methylpyridazin-3-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-fluoro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
(1S,4S)-5-(furan-3-ylmethyl)-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N-{2-methyl-4-[2-(1H-1,2,3,4-tetrazol-1-yl)acetamido]phenyl}pentanamide
2-methyl-4-{5-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]furan-2-yl}but-3-yn-2-ol
3-(2-ethylbutyl)-8-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(3-chlorophenyl)ethyl]-1-methylpiperidine-2-carboxamide
1-[(2S,4R)-4-[(4-methoxyphenyl)sulfanyl]-1-{[4-(trifluoromethoxy)phenyl]methyl}pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
2-cyclopropyl-6-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-1,3-benzoxazole
[1-(1-{[4-(5-methylfuran-2-yl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methanol
methyl N-{[(2S,4S)-4-fluoro-1-{2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetyl}pyrrolidin-2-yl]methyl}carbamate
{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
3-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyrimidin-2-amine
5-(dimethylamino)-2-(2-oxo-2-{2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}ethyl)-2,3-dihydropyridazin-3-one
N-cyclopentyl-3-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
2-[9-(5-acetylpyridin-2-yl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetic acid
N-[(3S)-1-benzylpiperidin-3-yl]-4-(pyridin-2-yl)pyrimidin-2-amine
N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2-(pyridin-2-yl)pyrimidine-5-carboxamide
1-(2-methoxyethyl)-2-oxo-3-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
1-(1-cyclopropylethyl)-5-(2-fluorophenyl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
1-(2-methanesulfonylethyl)-4-[3-(1H-pyrazol-4-yl)benzoyl]piperazine
6-[(3-fluorophenyl)methoxy]-4-(2-methoxyacetyl)-1-(2-phenylethyl)-1,4-diazepan-2-one
4-(1H-imidazol-1-yl)-1-[(4-methylthiophen-2-yl)sulfonyl]piperidine-4-carboxylic acid
4-[5-(methoxymethyl)thiophene-2-carbonyl]-1λ6-thiomorpholine-1,1-dione
2-amino-6-cyclobutyl-4-{3-[(dimethylamino)methyl]-4-methoxyphenyl}pyridine-3-carbonitrile
2,6-dihydroxy-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]benzamide
7-(2,6-dimethylquinoline-4-carbonyl)-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-1-[2-(thiophen-2-yl)ethyl]urea
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl){[2-(propan-2-yl)pyrimidin-5-yl]methyl}amine
2-methoxy-1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-2-(morpholin-2-yl)acetamide
4-(benzyloxy)-1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}piperidine
3-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-6-phenylpyridazine
N-cyclopropyl-N-[(7-methoxy-2-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}quinolin-3-yl)methyl]-3-methylthiophene-2-carboxamide
methyl 2-hydroxy-5-[6-oxo-1-(pentan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]benzoate
N-(2,3-dihydro-1H-inden-1-yl)-3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
methyl (2R,4S)-4-hydroxy-1-[(4-methoxynaphthalen-1-yl)methyl]piperidine-2-carboxylate
6-{3-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-3-oxopropyl}-2,3,4,5-tetrahydropyridazin-3-one
3-{5-[2-(4,6-dimethyl-1-benzofuran-3-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,2,8-trimethylquinoline-4-carboxamide
1-{[(3R,4R)-1-(5-chloro-3-fluoropyridin-2-yl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
N-(butan-2-yl)-7-(pyridine-4-amido)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
2-methyl-5-{[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-pyrrole-3-carbonitrile
1-{2-[1-(2,3-dihydroxypropyl)piperidin-4-yl]ethyl}pyrrolidin-2-one