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[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
(4aR,8aR)-4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-octahydro-2H-1,4-benzoxazine
3-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-6-methyl-1,2-dihydropyridin-2-one
4-({2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidin-1-yl}sulfonyl)morpholine
1-(1-methyl-1H-pyrazole-3-carbonyl)-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-ethyl-2-fluoro-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-5-sulfamoylbenzamide
7-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
5-(3-ethoxypropanoyl)-1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-{4-[1-(2,2,2-trifluoroethyl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}piperidine
(1S,3R)-3-[(dimethylsulfamoyl)amino]-N-[2-(5-methylthiophen-2-yl)ethyl]cyclopentane-1-carboxamide
2-[2-({3-[(pyridin-4-ylmethyl)carbamoyl]piperazin-1-yl}methyl)phenoxy]acetic acid
2-[3-(ethylsulfanyl)phenyl]-3-(piperidine-1-carbonyl)pyridine
4-benzyl-3-ethyl-1-(2-methoxy-5-methylbenzoyl)-1,4-diazepan-5-one
2-{2-[1-(2-hydroxybutyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2,3-dihydro-1H-isoindol-1-one
5-acetyl-N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}thiophene-3-carboxamide
3-(9H-purin-6-yl)phenol
1-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidin-1-yl)-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-methylacetamide
2-amino-3-ethyl-N-[(5-phenylfuran-2-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
[(5-ethylpyridin-2-yl)methyl](methyl)[(1-methyl-1H-indol-6-yl)methyl]amine
1-(4-ethenylphenyl)-3-(2-hydroxyethyl)-3-[(trimethyl-1H-pyrazol-4-yl)methyl]urea
2-{1-[(5-methylfuran-2-yl)methyl]-4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl}ethan-1-ol
4-(4-chlorophenyl)-N-[2-methoxy-1-(pyridin-2-yl)ethyl]butanamide
6-chloro-2-{[1-(4-chloro-2-methylphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydropyridazin-3-one
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)oxane-4-carboxamide
7-(3-{[2-(dimethylamino)ethyl](methyl)amino}piperidine-1-carbonyl)quinolin-8-ol
3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]propanamide
1-{3,5-dimethyl-4-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]-1H-pyrrol-2-yl}ethan-1-one
4-{1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}benzoic acid
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[4-(difluoromethoxy)benzoyl]piperidine
4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-propylfuran-2-yl)methyl]piperidine
3-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-1-(pyrrolidin-1-yl)propan-1-one
2-[2-(morpholin-4-ylmethyl)phenyl]pyridine-4-carboxamide
1-(2-ethoxypyridine-3-carbonyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
3-cyclopropyl-1-(3,4-difluorophenyl)-5-[(propan-2-ylsulfanyl)methyl]-1H-1,2,4-triazole
2-[1-(2-methylpropyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl][(4-{[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]amine
(3aS,6aS)-2-cyclohexyl-5-(pyridin-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(6-cyclopropylpyrimidin-4-yl)-4-(furan-3-carbonyl)-1,4-diazepan-6-ol
N-cyclopropyl-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-5-methylthiophene-2-carboxamide
N-(1-benzothiophen-5-ylmethyl)-2-methanesulfonamidoacetamide
{4-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]-1,4-oxazepan-6-yl}methanol
methyl 2-[(4aR,8aR)-6-(3-methoxybenzoyl)-decahydro-1,6-naphthyridine-1-carbonyl]benzoate
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-3-ylmethoxy)-4-(quinoxalin-5-ylmethyl)-1,4-diazepan-2-one
1-(3-{[(dimethylsulfamoyl)amino]methyl}piperidin-1-yl)-4-(4-fluorophenyl)butane-1,4-dione
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-5,6-dimethyl-N-(2-methylpropyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
4-(oxan-4-yl)-N-(trimethyl-1H-pyrazol-4-yl)piperazine-1-carboxamide
4-[(4-chlorophenyl)methyl]-1-(3-fluoropyridin-2-yl)piperidine-4-carboxylic acid
3-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}pyridin-2-amine
3-(5-chloro-2-methoxyphenyl)pyridin-4-amine