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2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-2,3-dihydro-1H-indene-2-carboxamide
N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-2-carboxamide
1-[(3,4-difluorophenyl)methyl]-4-(2-methylpyridin-4-yl)-1,4-diazepane
3-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl}-1,2-dimethyl-1H-indol-5-ol
4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}benzamide
2-(4-{2-[(2-methoxyethyl)amino]-1-methyl-1H-1,3-benzodiazole-5-carbonyl}morpholin-3-yl)acetamide
5-ethyl-N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]pyrimidin-2-amine
N,6-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-propylpyrimidin-4-amine
3-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}pyridin-2-ol
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylisoquinoline-3-carboxamide
1-({5-[1-(2-ethylbutyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)-4-methylpiperazine
5-methyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1H-1,3-benzodiazole-2-carboxamide
1-(cyclopropylmethyl)-5-(4-methyl-1H-imidazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-{3-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-1H-pyrazol-1-yl}-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
N-butyl-3-({4-[(3-methoxyphenyl)methyl]piperazin-1-yl}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
3-benzyl-1-methyl-8-[(3-methylquinoxalin-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S)-1-ethyl-4-[5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carbonyl]-3-methylpiperazin-2-one
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
1-[5-({[2-(2-chlorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(diethylamino)propan-2-ol
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-2-fluoro-N-methyl-5-sulfamoylbenzamide
ethyl 5-benzoyl-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}-3-propoxypiperidine
2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-[2-(1,3-thiazol-4-yl)ethyl]acetamide
ethyl 1-(2-methoxyethyl)-5-(3-phenyl-1H-pyrazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-3-phenoxypropan-1-one
2-{[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-4,6-dimethylpyrimidine
(2R)-2-amino-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}propanamide
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[2-(trifluoromethyl)morpholin-4-yl]ethan-1-one
6-methyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}pyridine-3-carboxamide
4-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2-[(3-fluorophenyl)methyl]morpholine
N-[3-(1,3-benzoxazol-2-yl)propyl]-2-cyclopropyl-4-hydroxypyrimidine-5-carboxamide
1-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]-4-phenylbutane-1,2-dione
2-(2-ethyl-1H-imidazol-1-yl)-1-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethan-1-one
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
2-[3-(2-ethylbutyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl]benzonitrile
4-methyl-5-{1-[2-(thiophen-2-yl)ethyl]-1H-pyrazol-3-yl}-N-[(2,4,5-trimethoxyphenyl)methyl]-1,3-thiazol-2-amine
1-[2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]piperidin-4-ol
N-(3-{[(1-hydroxybutan-2-yl)carbamoyl]methoxy}phenyl)propanamide
1-[4-({3-[(3,4-difluorophenyl)amino]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
3-amino-N-({1-[(2-cyanophenyl)methyl]pyrrolidin-3-yl}methyl)benzamide
2-[4-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)morpholin-3-yl]-N-phenylacetamide
(4-{[(1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)amino]methyl}oxan-4-yl)methanol
(3R,4S)-4-cyclopropyl-N,N-dimethyl-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]pyrrolidin-3-amine
3,4-dimethyl-N,N-bis(1,3-oxazol-4-ylmethyl)-5-sulfamoylbenzamide
1-(2-{2-[(4,4-difluoropiperidin-1-yl)methyl]phenoxy}ethyl)-4-methylpiperazine
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methylpiperidine-2-carboxamide
(3R,4R)-3-cyclobutyl-1-(1H-imidazol-2-ylmethyl)-4-methylpyrrolidin-3-ol
(2S)-2-(2,3-difluorophenyl)-2-[(8-fluoroquinolin-2-yl)formamido]acetic acid
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
2-[(3-{[(2E)-3-phenylprop-2-en-1-yl](prop-2-en-1-yl)carbamoyl}phenyl)amino]acetic acid