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N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
8-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[1-(3-methylbut-2-en-1-yl)-4-[(3-methylthiophen-2-yl)methyl]piperazin-2-yl]ethan-1-ol
4-{[(4-methyl-1H-imidazol-5-yl)methyl]amino}-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
3-ethyl-3-[(3S,4R)-4-hydroxyoxolan-3-yl]-1-[4-(trifluoromethyl)phenyl]urea
5-chloro-2-{4-[(2,6-difluoro-4-methoxyphenyl)methyl]piperazin-1-yl}pyrimidine
3-(azepane-1-sulfonyl)-5-(3,5-dimethoxyphenyl)benzoic acid
[(2S)-1-(4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)pyrrolidin-2-yl]methanol
ethyl 4-[1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-3-yl]piperazine-1-carboxylate
2-methoxy-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]pyridine-3-carboxamide
N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
5-{[(pyrimidin-2-yl)amino]methyl}adamantan-2-ol
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1H-indazole-3-carbonyl)piperidin-3-ol
N-[2-(4-ethoxyphenyl)ethyl]-1-(pyridin-2-yl)piperidine-3-carboxamide
6-{2-[3-oxo-3-(pyrrolidin-1-yl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}pyridine-3-carbonitrile
1-{[benzyl(1,3-thiazol-2-ylmethyl)carbamoyl]methyl}piperidine-4-carboxamide
ethyl 4-[(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-1-oxo-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-5-yl]-1H-pyrazole-3-carboxylate
N3-cycloheptyl-N5-[2-methyl-2-(morpholin-4-yl)propyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
5-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-N-ethylpyrimidin-2-amine
5-{3-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-3-oxopropyl}-5-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-2-one
4-(4-fluorophenyl)-4-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]butanamide
3-(2-methoxyphenyl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1H-pyrazole-5-carboxamide
1-methyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
5-ethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1,3,4-oxadiazol-2-amine
N-[3-(1H-imidazol-1-yl)propyl]-2,2-dimethyl-N-(pyridin-3-ylmethyl)oxane-4-carboxamide
3-[2-(4-fluorophenyl)ethyl]-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidine
2-chloro-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]pyridine-4-carboxamide
1-(3-{3-[(3-methoxypyrrolidin-1-yl)methyl]phenoxy}propyl)piperidine
methyl({[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl})[1-(1,3-thiazol-2-yl)ethyl]amine
1-methyl-4-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carbonyl)piperazine
3-{[1-(hydroxymethyl)cyclobutyl]methyl}-1-(5-methoxy-2-methylphenyl)-3-methylurea
2-methyl-6-{1-[1-(propan-2-yl)piperidine-3-carbonyl]piperidin-4-yl}pyrimidin-4-ol
2-[4-(4-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-3-carboxamide
4-cyclopropyl-6-{4-[2-(pyrrolidin-1-yl)ethyl]piperazin-1-yl}pyrimidine
N-{2-[benzyl(methyl)amino]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl}-2-(dimethylamino)acetamide
7-(cyclobutylmethyl)-2-(5-fluoro-1-methyl-1H-indole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[1-(pyridin-3-yl)ethyl]benzamide
methyl[3-(methylsulfanyl)propyl][(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amine
7-cyclopentyl-2-[3-(pyrazin-2-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
4-{4-[benzyl(methyl)amino]piperidin-1-yl}-5-methylpyrimidin-2-amine
9-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
methyl 3-benzamido-6-{[(2-methoxy-2-oxoethyl)(methyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
(1R,4S)-N-[3-(1,3-benzoxazol-2-yl)propyl]-1,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-4-carboxamide
3-{[2-(pyridin-3-yl)morpholin-4-yl]methyl}benzoic acid
1-{[5-(3-hydroxy-4-methylbenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}piperidin-3-ol
1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-(4,7-dimethylquinazolin-2-yl)-N-(2-methylbutyl)azepan-4-amine
3-[2-(3,4-difluorophenyl)ethyl]-1-(ethanesulfonyl)piperidine