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(1R,9aR)-N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-octahydro-1H-quinolizine-1-carboxamide
N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
3-({[(2,6-dimethylpyridin-4-yl)methyl]amino}methyl)-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
N-[1-(4-chlorophenyl)ethyl]-3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzamide
methyl 2-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanoate
8-{[3-(4-chlorophenoxy)phenyl]methyl}-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[3-(3-{furo[3,2-c]pyridin-4-yl}phenyl)-1H-pyrazol-1-yl]-N-methylacetamide
4-[5-methyl-4-(thiophen-2-yl)-1H-imidazol-2-yl]-1-(2-methylpropyl)pyrrolidin-2-one
2-amino-4-(2-fluoro-4-methylphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[(3-methoxyphenyl)methyl]-3-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-3-yl)propanamide
2-[1-(2-phenylethyl)-4-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol
N-methyl-3-(4-methyl-1H-pyrazol-1-yl)-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}propanamide
1-(5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carbonyl)-4-(propan-2-yl)piperazine
7-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(3-methoxypropyl)acetamide
3-[(4aR,7aS)-4-[(2-chlorophenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
N-ethyl-N-(4-hydroxybutyl)-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
1-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-4-(pyridin-4-yl)piperazine
5-{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]methyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(cyclohex-3-ene-1-carbonyl)-4-(4-methylphenoxy)piperidine-4-carboxylic acid
3-(3-fluorophenyl)-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]benzamide
2-(1-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1,3-benzothiazole
2-ethyl-8-[4-(1H-1,2,4-triazol-3-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[(1-{[(1-methyl-1H-pyrazol-4-yl)carbamoyl]methyl}pyrrolidin-3-yl)methyl]benzoic acid
3-({[7-(4-chlorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
1-[3-(4-phenylbenzoyl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
3-[2-(azocan-1-yl)-2-oxoethyl]-4-(pyridin-2-ylmethyl)piperazin-2-one
3-(2-methoxyphenyl)-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]propanamide
N-(2-fluorophenyl)-4-(4-methoxyphenyl)-2-methyl-5-oxopiperazine-1-carboxamide
4-ethyl-3-{1-[4-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(3R,4R)-1-[(2-methoxynaphthalen-1-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
N-[(1S)-2-(1H-imidazol-4-yl)-1-[1-phenyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl]acetamide
2-({3-[benzyl(methyl)amino]piperidin-1-yl}methyl)-4-methoxyphenol
5-cyclobutanecarbonyl-1'-[(3-fluorophenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl 3-{1-[2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)acetyl]piperidin-4-yl}propanoate
(3S,4R)-1-(dimethyl-1,3-thiazole-5-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
3-({3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyridin-2-amine
(2S)-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(methylamino)propanamide
1-{1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]azetidin-3-yl}piperidine
2-methoxy-N-{1-[1-(3-methylbut-2-enoyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
5-cyclohexaneamido-1-(2-methoxyethyl)-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole-7-carboxamide
2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propan-1-amine
3-(2-methoxyethyl)-1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)piperidine-3-carboxylic acid
5-(3,4-dimethoxyphenyl)-3-{octahydropyrrolo[1,2-a]piperazin-2-yl}-1,2,4-triazine
4-(3-methoxy-5-methylthiophene-2-carbonyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
1-(cyclopropylmethyl)-4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazine
3-(3-hydroxy-3-methylbutyl)-N-[(1R,2S)-2-phenylcyclopropyl]benzamide
2,6-dimethyl-N-[1-(methylcarbamoyl)cyclohexyl]imidazo[1,2-a]pyridine-3-carboxamide
5-{1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}-3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]imidazolidine-2,4-dione