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N-[2-(dimethylamino)ethyl]-3-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]propanamide
1-{1-[1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}cyclopentan-1-ol
4-(4-fluorophenyl)-N-methyl-4-oxo-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}butanamide
2-(dimethyl-1,3-thiazol-4-yl)-N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
4-[(4-fluorophenyl)methyl]-1-[(3-methoxyphenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-methyl-N-{[6-(morpholin-4-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-1,3-thiazole-4-carboxamide
(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-7-[(thiophen-2-ylmethyl)amino]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
methyl(2-methylpropyl)[(5-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]amine
6-methyl-2-{1-methyl-2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-yl}pyridine-3-carboxamide
2-fluoro-N-{3-[methyl(phenyl)amino]propyl}-5-sulfamoylbenzamide
8-methyl-2-[2-(morpholin-4-yl)pyridine-3-carbonyl]-2,8-diazaspiro[4.5]decane
(1S,5R)-6-benzyl-3-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
dimethyl({5-[1-(pyridine-2-carbonyl)piperidin-4-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amine
1-(propan-2-yl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]piperidine-4-carboxamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)piperidin-2-one
3-(4-chlorophenyl)-1-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidine
1-(5-chloropyridin-2-yl)-4-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine
3-{1-[1-(3-aminopropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea
[1-(3,5-dimethylbenzoyl)-4-(2-phenoxyethyl)piperidin-4-yl]methanol
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[3-(methylsulfanyl)propyl]benzamide
1-[4-(1-hydroxy-2-methylpropyl)piperidin-1-yl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propan-1-one
2-(4-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-1,3-benzothiazole
({4-cyclopropyl-5-[1-(2-phenylethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
4-(piperidin-3-yl)-N-[2-(pyridin-4-yl)ethyl]benzamide
1-methyl-3-(2-methylpropyl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1H-pyrazole-5-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-{1-[(1-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-2-yl}-1,3-thiazole
1-methyl-4-(1-{1-[4-(pyrrolidin-1-yl)benzoyl]piperidin-4-yl}ethyl)piperazine
1-[4-({[(3-ethyl-1,2-oxazol-5-yl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
1-ethyl-3-[8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]piperidine
3-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]-1-[2-(1,3,4-oxadiazol-2-yl)phenyl]urea
9-(but-3-yn-1-yloxy)-4-(2-methoxybenzoyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-{1-[3-(1H-pyrazol-1-yl)propanoyl]pyrrolidin-2-yl}-N-(pyridin-2-yl)thiophene-2-carboxamide
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3-[2-(4-fluorophenyl)ethyl]piperidine
2-methyl-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
[2-(cyclohex-1-en-1-yl)ethyl]({[6-(thiophen-3-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})amine
2-(1-benzylpiperidin-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
3-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-1-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}urea
2-[1-(3-methylbut-2-en-1-yl)-4-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperazin-2-yl]ethan-1-ol
2-amino-4-[1-(2-methylpropyl)-1H-indol-3-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-(3-hydroxy-3-phenylpropyl)-N,3-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1H-indole-5-carbonyl)piperidin-3-ol
6-methyl-2-[(2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-oxoethyl)sulfanyl]-3,4-dihydropyrimidin-4-one
1-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]azocane
4-[4-ethyl-6-(pyridin-4-yl)pyrimidin-2-yl]morpholine
8-(5-chloro-2-methoxybenzoyl)-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2-{4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,2-oxazole-3-carbonyl)piperidine
1-(propan-2-yl)-N-[2-(4-sulfamoylphenyl)ethyl]piperidine-3-carboxamide