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1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]azetidin-3-ol
4-{2-[1-benzyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]phenyl}morpholine
8-acetyl-2-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
6-(2-aminoethyl)-2-(3-{[(2H-1,3-benzodioxol-5-ylmethyl)(methyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
(3ar,6ar)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-(furan-3-ylmethyl)-N-methyl-1-[3-(1H-pyrazol-5-yl)phenyl]piperidin-4-amine
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-(1-ethylpiperidin-4-yl)acetamide
5-({5-[3-(ethoxymethyl)-4-methoxyphenyl]-4-phenyl-1H-imidazol-1-yl}methyl)-1H-1,2,4-triazole
N-ethyl-N-(2-methylprop-2-en-1-yl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
1-[(2E)-3-phenylprop-2-en-1-yl]-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-N'-(4-methylphenyl)propanediamide
2-(dimethylamino)-7-(5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-cyclohexyl-4-(2-oxo-1-phenylpyrrolidine-3-carbonyl)piperazin-2-one
5-acetyl-N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]thiophene-3-carboxamide
4-{1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}morpholine
6-methyl-2-(2-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)-3,4-dihydropyrimidin-4-one
2-[4-({4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenoxy]ethan-1-ol
4-[1-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)piperidin-3-yl]benzoic acid
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-4-methylphenyl)urea
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-(morpholin-4-yl)ethan-1-one
4-{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}thiomorpholine
2-{[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
[(3R,4R)-1-[(4-fluoro-2-methylphenyl)methyl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
1-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-3-propylurea
5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)-N-[(3-methylpyridin-2-yl)methyl]pyridin-2-amine
5-{2-[4-(adamantan-1-yl)piperazin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
[(1-ethyl-1H-pyrazol-4-yl)methyl](furan-3-ylmethyl)(2-methylpropyl)amine
(3S)-3-ethyl-4-{[5-(2-methyl-1,3-thiazol-4-yl)thiophen-2-yl]sulfonyl}morpholine
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-ethyl-N-(pyridin-3-ylmethyl)-1,2-oxazole-5-carboxamide
ethyl 3,5-dimethyl-4-{5-oxo-1,4,9-triazaspiro[5.5]undecane-9-carbonyl}-1H-pyrrole-2-carboxylate
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-hydroxy-2-[(phenylsulfanyl)methyl]pyrimidine-5-carboxamide
2-(2-chlorophenoxy)-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
N-[(8-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]acetamide
1-{1-tert-butyl-3-[(2,6-dichlorophenyl)methyl]-1H-1,2,4-triazol-5-yl}cyclopropane-1-carboxamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[(4-methylphenyl)amino]-2-phenylpropanamide
(3S,4S)-3-hydroxy-4-{2-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1H-imidazol-1-yl}-1λ6-thiolane-1,1-dione
N-(2,3-dihydro-1H-inden-5-yl)thiomorpholine-4-carboxamide
1-{4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}-3-(thiolan-3-yl)urea
[2-(3-methyl-3-phenylpiperidin-1-yl)pyridin-4-yl]methanol
5-{5-[(1-methyl-1H-imidazol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-N-propylpyrimidin-2-amine
N,N-dimethyl-2-(4-{[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperazin-1-yl)acetamide
N-methyl-1-[1-(3-phenylpropyl)piperidin-4-yl]-N-(1H-pyrazol-5-ylmethyl)piperidine-4-carboxamide
3-(1H-indol-3-yl)-1-[3-(3-methoxybenzoyl)piperidin-1-yl]propan-1-one
7-(furan-2-ylmethyl)-N-methyl-N-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
6-oxo-N-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}-1,4,5,6-tetrahydropyridazine-3-carboxamide
1-(3-{[4-(trifluoromethyl)pyrimidin-2-yl]amino}propyl)pyrrolidin-2-one
1-acetyl-N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)piperidine-4-carboxamide
3-benzoyl-1-(1-phenylpyrrolidin-3-yl)piperidine
(3R,4S)-1-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3,4-dimethylpiperidin-4-ol
1-{4-[(3-ethoxypropyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one