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N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]acetamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-N,5-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
4-{6-[4-(2-methylphenyl)piperazin-1-yl]pyrimidin-4-yl}morpholine
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-3-(2,5-dioxoimidazolidin-4-yl)propanamide
4-{[(2-methoxyphenyl)methyl]amino}-N,5-dimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
6-{2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
(benzylsulfamoyl)(ethyl)[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]amine
10-methoxy-5-[4-(piperidin-3-yl)benzoyl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
methyl N-{2-[(1S,5R)-6-benzyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}carbamate
4-[(1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}pyrrolidin-3-yl)methyl]benzoic acid
(3S,4S)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(piperidin-1-yl)pyrrolidin-3-ol
N-(1-ethylcyclopropyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)imidazo[1,2-a]pyrimidine-2-carboxamide
N-[(1-methylpyrrolidin-3-yl)methyl]-2-(thiophene-2-sulfonamido)acetamide
2-(3-{[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]methyl}phenyl)-6-methyl-3,4-dihydropyrimidin-4-one
2-(4-acetyl-1,4-diazepan-1-yl)-2-(2,3-dimethoxyphenyl)acetic acid
N-benzyl-N,6-dimethyl-2-(4-methylphenoxymethyl)-1-[2-(morpholin-4-yl)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-{[2-(dimethylamino)-7-(methylsulfanyl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)cyclopropanecarboxamide
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-[2-(2-methoxyphenyl)ethyl]pyrrolidin-2-one
5-(3-acetylphenyl)pyridine-3-carboxamide
3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[3-(methylsulfanyl)propyl]propanamide
3-methyl-6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyridazine
N-(2,2-dimethylpropyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
4-benzyl-3-ethyl-1-[(1-methyl-1H-imidazol-2-yl)methyl]-1,4-diazepan-5-one
2-{6-[(dimethylamino)methyl]-1,4-oxazepan-4-yl}-N-methylpyridine-3-carboxamide
2-(2-ethyl-1H-imidazol-1-yl)-1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
N-(1-benzothiophen-2-ylmethyl)-6-{[cyclohexyl(methyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
4-[3-(4-benzylpiperidine-1-carbonyl)piperidin-1-yl]-2-[(4-methyl-1,3-thiazol-2-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
5-fluoro-1,3-dimethyl-2-[4-(pyrimidin-2-yloxy)piperidine-1-carbonyl]-1H-indole
N-(2,5-dimethylphenyl)-3-[4-(pyridin-3-yloxy)piperidin-1-yl]propanamide
3-{[1-benzyl-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenol
N-[2-(2-fluorophenyl)ethyl]-2-oxa-7-azaspiro[4.5]decane-7-carboxamide
1-(methoxymethyl)-N-methyl-N-[(4-phenylphenyl)methyl]cyclobutane-1-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)amine
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)(pyridin-2-ylmethyl)amine
1-{3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}cyclopentan-1-amine
1-(2-hydroxyethyl)-N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
1-{4-[2-(4-methoxy-2,3-dimethylphenyl)-1H-imidazol-1-yl]butan-2-yl}-4-methylpiperazine
2-[4-(propan-2-yloxy)phenyl]-4-[1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]pyridine
4,6-dimethyl-5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazolo[3,4-b]pyridin-3-amine
(3R,5S)-N-cyclopropyl-5-(morpholin-4-ylmethyl)-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
2-(3-fluorophenyl)-N-({7-[(2,4,5-trimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
1-(2-ethoxyethyl)-2-oxo-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-(1H-pyrazol-1-yl)-N-[(1S,3S)-3-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}cyclopentyl]propanamide
4-(4-ethyl-6-{[1-(morpholin-4-yl)hex-5-en-2-yl]oxy}pyrimidin-2-yl)morpholine
1-(2-chloro-3-methylbenzoyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
3-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)-N-(1,2,4-thiadiazol-5-yl)benzamide