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3-(1,3-benzothiazol-2-yl)-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]propanamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-4-(piperidin-1-ylmethyl)benzamide
1-(4-chloro-1H-pyrazole-3-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(2S)-N-{[7-(1,3-benzothiazol-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-oxopyrrolidine-2-carboxamide
2-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
2-(2H-1,3-benzodioxol-5-yloxy)-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]propan-1-one
9-(2-hydroxyethyl)-1-methyl-4-{thieno[3,2-d]pyrimidin-4-yl}-1,4,9-triazaspiro[5.6]dodecan-10-one
(4aR,8aS)-1-[2-(4-methoxyphenyl)ethyl]-6-[(3-methylphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
N,N-dimethyl-5-({2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)pyrimidin-2-amine
3-(5-{7-methyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)-N-(propan-2-yl)propanamide
{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
1-cyclohexyl-4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]-1,4-diazepane
N-[(2,3-dimethoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)morpholine-2-carboxamide
N,8-dimethyl-3-({methyl[(methylcarbamoyl)methyl]amino}methyl)-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
(4aR,8aS)-1-[2-(3-methoxyphenyl)ethyl]-6-[4-(trifluoromethyl)benzoyl]-decahydro-1,6-naphthyridin-2-one
4-ethyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-1,2,3-thiadiazole-5-carboxamide
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)furan-2-carboxamide
2-(2-hydroxyethyl)-8-[(2-phenyl-1,3-thiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]acetic acid
(3S,4R)-1-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]-3-methoxypiperidin-4-amine
3-{2-[3-(methoxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-2,6,6-trimethyl-1-propyl-4,5,6,7-tetrahydro-1H-indol-4-one
3-({[(3S,4R)-4-hydroxyoxolan-3-yl](methyl)amino}methyl)-5,6,7-trimethoxy-1,2-dihydroquinolin-2-one
(1s,4s)-4-(4-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)cyclohexan-1-amine
(2,4,6-trimethyl-3-{[4-(oxolane-2-carbonyl)piperazin-1-yl]methyl}phenyl)methanol
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
4-{4-[4-(2-methoxyethyl)piperazine-1-carbonyl]-5-methyl-1H-pyrazol-1-yl}-3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaene
5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxamide
1-{1-[(2,4-difluorophenyl)methyl]-4-phenylpiperidin-4-yl}ethan-1-one
1-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}piperazine
N-(3,5-dimethoxyphenyl)-3-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-3-yl}propanamide
3-[(2R,3R,6R)-5-(2-methylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylthian-4-amine
3-(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-3-yl)-N-[(5-methylfuran-2-yl)methyl]propanamide
N-(4-methoxy-2-methylphenyl)-3-{1-[2-(methylsulfanyl)benzoyl]piperidin-3-yl}propanamide
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
3-{1-[1-(2,5-difluorobenzenesulfonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-1-ol
{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
N-[1-(3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]pyridin-2-amine
2-[4-(1,3-oxazol-5-yl)benzenesulfonyl]-2,7-diazaspiro[4.5]decane
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
3-[5-(methoxymethyl)-1-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]pyridine
5-cyclopropyl-4-{[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-methyl-1H-pyrazole
N-cyclopropyl-N-({4-[3-(dimethylamino)propoxy]phenyl}methyl)-4-methylbenzamide
({6-methyl-2-[(2-methylphenyl)methoxy]quinolin-3-yl}methyl)[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]amine
(4aS,8aR)-1-(3-methoxypropyl)-6-(1-propyl-1H-pyrazole-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]butanamide
3-(difluoromethoxy)-N-(5-oxo-1-phenylpyrrolidin-3-yl)benzamide
3-{5-[(3-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}urea
3-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[(5-methylthiophen-2-yl)methyl]amino)propan-1-ol