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[1-(2-{[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}ethyl)piperidin-2-yl]methanol
7-methoxy-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
3-[1-(1-methyl-1H-imidazol-2-yl)butyl]-1-[4-methyl-3-(2-oxopyrrolidin-1-yl)phenyl]urea
3-({4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)-1H-indole
N-[3-(pyridin-3-yloxy)propyl]-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)-1-[4-(thian-4-yl)piperazin-1-yl]propan-1-one
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
6-fluoro-3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,4-dihydroquinazolin-4-one
N-(2-methoxyethyl)-1-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
3-(2-methylphenoxymethyl)-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidine
4-(4-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}-2-oxopiperazin-1-yl)benzonitrile
3-[4-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)-1H-pyrazol-1-yl]propanoic acid
3-(2-fluoro-3-methoxyphenyl)pyrazolo[1,5-a]pyrimidine
2-acetyl-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]benzamide
2-methyl-5-{[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
(3R,9aR)-3-[(1S)-1-hydroxyethyl]-8-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-cyclopropyl-2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-4-carboxamide
1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
3-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propane-1,2-diol
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl)[(6-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
2-{[2-(adamantan-1-yl)-1,3-thiazol-4-yl]methyl}-5-(dimethylamino)-2,3-dihydropyridazin-3-one
2-cyclopropyl-8-[(3,4-dimethylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
methyl 2-(diethylsulfamoyl)-6-[4-(methoxycarbonyl)benzoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-ethyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
N1-(3-methylpyridin-4-yl)-N2-(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)ethane-1,2-diamine
2-(2-{[cycloheptyl(ethyl)amino]methyl}phenyl)-5,6-dimethyl-3,4-dihydropyrimidin-4-one
(1R,2S,9R)-11-(quinoxalin-2-yl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
3-[(4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperazin-1-yl)methyl]phenol
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-(2-phenoxyethyl)-decahydroisoquinoline
(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-[(4-methoxyphenyl)methyl]piperidin-4-yl)methanol
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-(4-phenylphenyl)propan-1-one
1-{2-[({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)amino]ethyl}imidazolidin-2-one
1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-[2-({1,9-dioxaspiro[5.5]undecan-4-yl}amino)ethyl]pyridine-3-carboxamide
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl](methyl)[(5-methylfuran-2-yl)methyl]amine
2-chloro-N-(1-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-{[7-(1,3-benzothiazol-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-3-carboxamide
2-(2-{2-[2-(dimethylamino)ethyl]piperidin-1-yl}-2-oxoethyl)-3-phenylcyclopent-2-en-1-one
N-(4-methyl-4-phenylpentan-2-yl)-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
2-(4-amino-3-fluorophenyl)-2-[4-carbamoyl-4-(piperidin-1-yl)piperidin-1-yl]acetic acid
2-{4-[(3,3-difluoropiperidin-1-yl)methyl]phenyl}-6-methyl-3,4-dihydropyrimidin-4-one
1-[cyclohexyl(methyl)amino]-3-(3-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
2-(3-methyl-1,2-oxazol-5-yl)-N-[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]acetamide
3-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
2-{5-[(4,5-dimethyl-1H-imidazol-1-yl)methyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}acetic acid
5-(2-{3,9-diazaspiro[5.5]undecan-3-yl}-2-oxoethyl)-2-methyl-3,4-dihydropyrimidin-4-one
3-[5-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]-5-[2-(piperidin-2-yl)ethyl]phenol