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3-chloro-5-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-{2-[3-(pyridin-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
1-[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-5-one
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(1,3-dihydroxypropan-2-yl)acetamide
(1R,5R)-6-(cyclopropylmethyl)-3-(5,6-dimethylpyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonane
[2,4,6-trimethyl-3-({[2-(1H-1,2,4-triazol-1-yl)propyl]amino}methyl)phenyl]methanol
(2S,4S)-4-amino-1-hexanoyl-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[(2-ethoxyphenyl)methyl]-N-ethyl-3-(thiophen-3-yl)propanamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-(oxan-3-ylmethyl)benzamide
1-[(2,3-dioxo-1,2,3,4-tetrahydroquinoxalin-6-yl)sulfonyl]-3-propylpiperidine-3-carboxylic acid
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-1-[(3,4-dimethoxyphenyl)methyl]-N-[2-(1-methylpyrrolidin-2-yl)ethyl]piperidine-3-carboxamide
(8aS)-2-{[2-(3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
3-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1-benzofuran-4-one
3-methyl-5-(1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}pyrrolidin-2-yl)-1H-1,2,4-triazole
3-{[4-(cyclopropylmethyl)piperazin-1-yl]methyl}-1-[(2,3-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
N-(2,6-dimethylphenyl)-3-(2-hydroxy-2-phenylpropanamido)benzamide
(1S,4S)-2-(2-fluorophenyl)-5-[(8-methoxyquinolin-2-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3R,4R)-4-(morpholin-4-yl)-1-[4-(trifluoromethyl)pyridin-2-yl]piperidin-3-ol
(3aR,6aR)-2-acetyl-5-[(1-ethyl-1H-imidazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{4-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
4-{1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-3-yl}benzoic acid
(1R,5S)-3-benzyl-6-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-[4-(cycloheptylcarbamoyl)piperidin-1-yl]-2-(4-fluoro-3-methylphenyl)acetic acid
1-{1-[2-(5-ethyl-1-benzofuran-3-yl)acetyl]piperidin-3-yl}pyrrolidin-2-one
4-[(2,4-difluoro-3-methoxyphenyl)methyl]-3-ethyl-1-methylpiperazin-2-one
4-[4-(benzyloxy)piperidine-1-carbonyl]-1-cyclopropylpyrrolidin-2-one
1-[2-(2H-1,3-benzodioxol-5-yl)pyrimidin-4-yl]piperidin-3-ol
dimethyl(2-{1-[(1-methyl-1H-imidazol-5-yl)methyl]piperidin-2-yl}ethyl)amine
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-{[1-(2-chlorophenyl)-3-cyclopentyl-1H-1,2,4-triazol-5-yl]methyl}morpholine
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(1-methylpiperidin-4-yl)-decahydro-1,6-naphthyridin-2-one
N-[(2-ethoxypyridin-3-yl)methyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-(3-benzyl-1H-pyrazol-5-yl)-1-[(2R)-oxolane-2-carbonyl]piperidine
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-N5-(2-phenylethyl)piperidine-3,5-dicarboxamide
6-[(3,4-dimethoxyphenyl)methyl]-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}(1,2-oxazol-3-ylmethyl)amine
7-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
6,7-dimethoxy-2-(2-propyl-1,3-thiazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline
1-(ethanesulfonyl)-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazine
8-{3-cyclopropyl-5-[2-(pyridin-3-yl)ethyl]-1H-1,2,4-triazol-1-yl}quinoline
1-(2-methoxy-4-{[(oxan-4-ylmethyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
6-(2-chlorophenyl)-N-(pyridin-4-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(2-{2-azabicyclo[2.2.1]heptan-2-yl}-2-oxoethyl)-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidine-2,5-dione
2-(1H-imidazol-1-yl)-1-(4-{[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
1-[1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
2-{3-[(3,4-dimethoxyphenyl)methyl]-5-(2-ethyl-4-methyl-1,3-oxazol-5-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-2-(propan-2-yloxy)propanamide
N-[4-(1H-indazol-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]piperidin-4-amine
3-methyl-1-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]but-2-en-1-one