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1-methyl-4-{3-[2-(oxolan-3-yl)-1H-imidazol-1-yl]propoxy}piperidine
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
2-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-[(1R,2R)-2-phenylcyclopropanecarbonyl]-7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(3,5-dimethylphenyl)-6-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(2,4-dimethoxyphenyl)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
2-[4-(2,1,3-benzothiadiazole-4-sulfonyl)morpholin-3-yl]-N-ethylacetamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(2-methoxyphenoxy)piperidin-1-yl]propan-1-one
2-(2-methylpropyl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
1-(4-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-4-oxobutyl)piperidin-2-one
N-(2-methoxy-5-methylphenyl)-3-[methyl(2-phenylethyl)amino]piperidine-1-carboxamide
(2R)-N-[1-(4-fluorophenyl)-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]oxolane-2-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]-1,4-diazepane
N'-{[1-(quinolin-8-ylmethyl)pyrrolidin-3-yl]methyl}ethanediamide
2-(morpholine-4-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
4-(methoxymethyl)-N,5-dimethyl-N-[(5-methylfuran-2-yl)methyl]-1,2-oxazole-3-carboxamide
4-[3-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)propyl]-1,3-thiazol-2-amine
1-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-3-yl}-4-(2-methoxyphenyl)piperazine
N-[3-(cyclohexyloxy)propyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
5-{[4-(2-methoxyethoxy)piperidin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
5-[butyl(methyl)amino]-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[1-(pyrazin-2-yl)propan-2-yl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-chloro-2-{[3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazin-1-yl]methyl}phenol
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-3,4,7-trimethyl-1H-indole-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-methyl-5-(oxolan-2-yl)thiophene-2-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-propyl-1,3,4-thiadiazol-2-amine
(2E)-N-cyclopentyl-N-{[3-methoxy-4-(oxan-2-ylmethoxy)phenyl]methyl}-3-(thiophen-2-yl)prop-2-enamide
4-(hydroxymethyl)-1-[4-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)benzoyl]piperidin-4-ol
N4-methyl-N4-[(2-phenyl-1,3-thiazol-4-yl)methyl]pyrimidine-2,4,6-triamine
5-(5-chloro-2-methoxyphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-{5-[(4-cyclohexyl-3-oxopiperazin-1-yl)methyl]-2-methoxyphenoxy}acetic acid
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-methyl-3-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}urea
3-[2-(1-methylpiperidin-2-yl)ethyl]-3H,4H-pyrido[4,3-d]pyrimidin-4-one
methyl[(3-methylthiophen-2-yl)methyl]{[5-(pent-2-yn-1-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}amine
(4aR,6R,8aS)-8a-(methoxymethyl)-2-[(5-methylthiophen-2-yl)methyl]-6-(morpholin-4-yl)-decahydroisoquinoline
3-[2-(azepan-1-yl)-2-oxoethyl]-1-(2-methoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
5-ethyl-N4-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}pyrimidine-2,4-diamine
(3S,4S)-1-(benzenesulfonyl)-4-[methyl(quinolin-6-ylmethyl)amino]pyrrolidin-3-ol
2-(4-{3-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}piperidin-1-yl)acetamide
6-[7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]pyridine-2-carboxamide
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4R)-1-(4-hydroxy-3-methoxybenzoyl)-4-phenylpyrrolidine-3-carboxylic acid
5-amino-4-phenyl-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-3-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(2-propyl-1,3-thiazol-4-yl)formamido]acetic acid
2-[(2-{1-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine
N-ethyl-2-methyl-N-(2-phenoxyethyl)furan-3-carboxamide
3-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfamoyl]benzoic acid
N-[3-(azepan-1-yl)propyl]-N-methyl-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
3-(2-oxoazepan-1-yl)-N-[(4-phenyloxan-4-yl)methyl]propanamide