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1-(2-chlorophenyl)-4-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperazin-2-one
3-({[2-(quinolin-8-yloxy)ethyl]amino}methyl)pyrrolidin-3-ol
6-fluoro-3-[1-(6-methylpyridin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]pyrrolidin-3-yl]methanol
1-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-3-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
N-(4H-1,2,4-triazol-4-yl)-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
5-ethyl-N-[(1R)-1-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-amine
N-(1-methylpiperidin-4-yl)-2-phenoxy-N-(2-phenylethyl)acetamide
N-({7-[3-(3-methoxyphenyl)propanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-4-carboxamide
3-{1-[3-(1H-imidazol-1-yl)propyl]piperidin-3-yl}benzoic acid
4-benzyl-1-{5-[(2E)-but-2-en-1-yl]-1,3,4-oxadiazole-2-carbonyl}piperidin-4-ol
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[(4-fluorophenyl)methyl]-5-methoxybenzamide
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[4-(1H-imidazol-1-yl)benzoyl]pyrrolidin-3-yl]methanol
methyl 5-({2-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]acetamido}methyl)furan-2-carboxylate
6-(2-aminoethyl)-2-[4-({methyl[3-(1H-pyrazol-1-yl)propyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
4-(3-ethyl-1H-pyrazole-4-carbonyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-2-(4-phenylpiperidin-1-yl)acetamide
4-{[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]methyl}benzoic acid
2-ethyl-N,4-dimethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1,3-thiazole-5-carboxamide
N,N-diethyl-2-({4-[2-(methylsulfanyl)acetyl]-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl}oxy)acetamide
3-chloro-N,6-dimethyl-N-(quinolin-5-ylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2,3-dimethyl-6-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetyl}-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]({[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})amine
[5-({[2-(azepan-1-yl)ethyl](propan-2-yl)amino}methyl)-2-methoxyphenyl]methanol
N,N-dimethyl-2-[(1S,5R)-6-{[3-(morpholin-4-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
3-(2-chlorophenyl)-4-(1H-imidazol-2-yl)-1-(4-methoxyphenyl)-1H-pyrazole
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl})amine
N'-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}ethanediamide
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
4-(3,6-dimethylpyrazin-2-yl)-2-[(4-phenylpiperidin-1-yl)methyl]phenol
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-methoxy-2-methylpropanamide
(1R,3S)-7-(1-benzoxepine-4-carbonyl)-7-azaspiro[3.5]nonane-1,3-diol
4-methyl-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
methyl 6-(cyclopropylmethyl)-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl 3-(cyclobutylmethoxy)-5-(5-oxo-1,4-diazepane-1-carbonyl)benzoate
1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S)-4-methanesulfonyl-2-{[3-(1H-pyrazol-1-yl)phenyl]formamido}butanoic acid
(1S,4S)-2-(2-chlorophenyl)-5-(2-methylpropyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
[(1-cyclohexylpiperidin-3-yl)methyl][(2,4-difluorophenyl)methyl](pyridin-3-ylmethyl)amine
3-(1,3-benzothiazol-2-yl)-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]propan-1-one
methyl (2S)-1-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)pyrrolidine-2-carboxylate
[3-(3-methylbut-2-en-1-yl)-1-(3-methylpyrazin-2-yl)piperidin-3-yl]methanol
1-(4-{3-[({[5-(2-methylpropyl)thiophen-2-yl]methyl}amino)methyl]pyridin-2-yl}piperazin-1-yl)ethan-1-one
9-(4-ethoxybenzoyl)-1-methyl-4-propyl-1,4,9-triazaspiro[5.5]undecane
1-(2-hydroxy-4-methylbenzoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[3-(piperidin-3-yl)benzoyl]-4-(pyridin-3-ylmethyl)piperazine
2-methyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-({4-[4-(3-methoxypiperidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)-6-methylpyridine