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N-[(3-chloro-1-benzothiophen-2-yl)methyl]-2-(2,5-dioxoimidazolidin-4-yl)-N-methylacetamide
2-(4-chlorophenyl)-4-[4-(1H-1,2,4-triazol-3-yl)benzoyl]morpholine
2-(2-chlorophenoxy)-1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
3-[1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-1-(pyrrolidin-1-yl)propan-1-one
2-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]methyl}-1-methyl-1H-1,3-benzodiazole
1,5-dimethyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
1-[2-(3-cyclohexylpyrrolidin-1-yl)-2-oxoethyl]-3-methoxy-1,2-dihydropyridin-2-one
1-[2-(2H-1,3-benzodioxol-5-yloxy)acetyl]-N-cyclopropylpiperazine-2-carboxamide
4-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}-1-phenyl-1H-1,2,3-triazole
2-methyl-6-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2,3-dihydropyridazin-3-one
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]pyrimidin-2-amine
7-(2-hydroxyethyl)-2-[2-(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
(8R,9aS)-8-hydroxy-2-[2-(1H-indol-1-yl)ethyl]-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(pyridin-3-yl)acetamide
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
dimethyl[3-(2-{1-[3-(pyrrolidin-1-yl)pyrazin-2-yl]piperidin-3-yl}-1H-imidazol-1-yl)propyl]amine
{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
6-fluoro-N-(isoquinolin-5-ylmethyl)-N-methyl-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(3S,4S)-1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-4-(piperidin-1-yl)pyrrolidin-3-ol
N-methyl-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
[(3R,4R)-1-(4-methanesulfonylbenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)-2,1,3-benzothiadiazole-4-sulfonamide
9-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-6-(4-methoxyphenyl)-6,9-diazaspiro[4.5]decan-7-one
1-cyclobutanecarbonyl-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]piperidine-4-carboxamide
6-(3-fluorophenyl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-3-[2-(methylsulfanyl)ethyl]-5-(oxan-4-yl)-1H-1,2,4-triazole
3-(4-methoxy-3,5-dimethylbenzoyl)-1-[(3,4,5-trimethoxyphenyl)methyl]piperidine
methyl 1-{3-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
N-(pyridin-2-ylmethyl)-1-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
2-{[4-(4-chlorophenyl)-5-[(propan-2-yloxy)methyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
(3S,4S)-4-cyclopropyl-1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]pyrrolidine-3-carboxylic acid
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(2-fluorophenyl)methyl]piperidine-3-carboxamide
1-[(4-acetamidophenyl)methyl]-4-(2-methylphenoxy)piperidine-4-carboxylic acid
(pentan-3-yl)[2-(pyridin-3-yloxy)propyl]amine
N-{[5-fluoro-7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methyl-1H-pyrazole-5-carboxamide
2-(3-fluoro-4-methoxyphenyl)-2-[4-(piperidine-1-carbonyl)piperidin-1-yl]acetic acid
4-[3-(5-methylfuran-2-yl)butyl]-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(4-ethyl-1H-pyrazol-5-yl)-1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperidine
4-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidine
(2S,4S)-4-amino-1-[(1-phenyl-1H-pyrazol-5-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-{5-[(3-ethyl-3-hydroxypiperidin-1-yl)methyl]-1,2,4-oxadiazol-3-yl}benzoic acid
N-[2-(3-methoxyphenyl)ethyl]-5-(4-methylpiperidine-1-carbonyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
1-benzyl-N-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-amine
(2-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)urea
N-(2-hydroxyethyl)-2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
3-{[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]methyl}-5-methanesulfonamido-N-phenylbenzamide
3-{5-[(2,3,5,6-tetrafluoro-4-methoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-(2-cyclopropylpyrimidin-5-yl)-4-(3,3-dimethylpyrrolidine-1-carbonyl)-7-fluoroquinoline
5-{imidazo[1,2-a]pyridin-6-yl}-4-phenyl-1H-imidazole