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2-methyl-5-[4-(5-methylpyridine-3-carbonyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
3-ethyl-1-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]piperidine-3-carboxylic acid
6-chloro-2-{2-oxo-2-[3-(4-phenylbenzoyl)piperidin-1-yl]ethyl}-2,3-dihydropyridazin-3-one
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-ethyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}acetamide
(1R,5S)-6-methyl-3-[2-(thiophen-2-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-3-propoxypiperidine
methyl({[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-{9-[2-(morpholin-2-yl)acetyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
5-chloro-N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)thiophene-2-carboxamide
9-[(dimethyl-1,3-thiazol-5-yl)methyl]-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{5-[(R)-cyclohexyl(hydroxy)methyl]-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl}acetic acid
3-[2-(1H-indol-1-yl)ethyl]-1-[4-(morpholin-4-ylmethyl)phenyl]urea
1-[(4-methyl-1H-imidazol-5-yl)methyl]-N-[3-(3-methylphenyl)phenyl]pyrrolidine-2-carboxamide
2-methyl-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)-1,3-thiazole-4-carboxamide
4-[2-(2-hydroxyethoxy)ethyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl){[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
3-butyl-4-ethyl-1-{2-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]-2-oxoethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 3-[4-(2-amino-3-cyano-6-cyclopentylpyridin-4-yl)-1H-pyrazol-1-yl]propanoate
N-benzyl-2-(dimethylamino)-N-[2-(dimethylamino)ethyl]-6-phenylpyridine-3-carboxamide
2-[3-oxo-9-(2-phenoxyethyl)-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
3-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenylurea
N3-(3-{[(2-methylphenyl)methyl]sulfanyl}propyl)piperidine-1,3-dicarboxamide
5-[(3-methoxyphenyl)methyl]-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
1-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]piperidine-3-carboxamide
1-(2-methoxyphenyl)-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazine
1-[(3-methylphenyl)methyl]-3-{pyrazolo[1,5-a]pyridin-3-ylmethyl}urea
1-{2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
2-(1H-indol-3-yl)-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)acetamide
3-({5-[1-(2,3-dihydro-1H-inden-2-yl)-1H-imidazol-2-yl]furan-2-yl}sulfanyl)-4-methyl-4H-1,2,4-triazole
(1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanol
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[methyl(1-methylpiperidin-4-yl)amino]ethan-1-one
7-[(2,3-difluorophenyl)methyl]-2-[3-(methylsulfanyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]-1-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]piperidine
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
2-(2H-1,3-benzodioxol-5-yl)-1-{4-[3-({methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenoxy]piperidin-1-yl}ethan-1-one
(4aR,8aR)-2-methanesulfonyl-7-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-decahydro-2,7-naphthyridin-4a-ol
3-({1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}methyl)-1-(4-methylphenyl)urea
3-{1-[2-(1H-1,3-benzodiazol-1-yl)acetyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
3-[3-(2-chlorophenyl)-N-methyl-3-phenylpropanamido]-N-methylpropanamide
1-(2-methoxyethyl)-4-{[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}pyrrolidin-2-one
1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2-amino-4-[5-chloro-2-(prop-2-en-1-yloxy)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-(cyclopropylmethyl)-3-{methyl[(1-methyl-5-oxopyrrolidin-3-yl)methyl]sulfamoyl}benzamide
2-({3-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-1,2-oxazol-5-yl}methyl)-1,2,3,4-tetrahydroisoquinoline
2-[(2-{[(1R)-1-phenylethyl]carbamoyl}phenyl)amino]acetic acid
N-(1,1-dioxo-1λ6-thian-4-yl)-N,1-dimethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide