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3-[(2-methoxyethyl)sulfamoyl]-5-(pyridin-3-yl)benzoic acid
7-hydroxy-4-{2-[3-(1H-imidazol-1-yl)propoxy]phenyl}-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
N-(2-methoxyethyl)-3,4,7-trimethyl-N-(pyridin-2-ylmethyl)-1H-indole-2-carboxamide
4,6-dimethyl-1-[2-({1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-yl}amino)ethyl]-1,2-dihydropyrimidin-2-one
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(3,4-dimethylphenyl)ethan-1-one
N2-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-N1-(3-methylpyridin-4-yl)ethane-1,2-diamine
(1-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}piperidin-4-yl)methanamine
4-(3-fluorophenyl)-N-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}benzamide
[4-(2-phenylethyl)-1-(3-phenylprop-2-yn-1-yl)piperidin-4-yl]methanol
3-{[cyclopropyl(3-methylpyridin-2-yl)methyl]amino}-N-(2-methylphenyl)propanamide
1,3-dimethyl-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1H-pyrazole-5-carboxamide
1-(2-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}-2-oxoethyl)-2-methyl-1H-indole-3-carbonitrile
1-(2-methyl-2,3-dihydro-1H-indol-1-yl)-2-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethane-1,2-dione
2-{[2-(phenylamino)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-{1-[1-(furan-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
4-({1-[(4-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)piperidine
4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-(1H-indazol-6-yl)piperazin-2-one
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-(propan-2-yl)acetamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3-ethyl-1,2-oxazole-5-carboxamide
(4aS,8aR)-6-(3-hydroxypyridine-2-carbonyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-(2,3-dihydro-1H-isoindol-2-yl)-2-(dimethylamino)-2-(2-fluorophenyl)ethan-1-one
6-(hydroxymethyl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]pyridine-2-carboxamide
3,3-dimethyl-1-{1-methyl-4-[(4-methyl-1,3-thiazol-2-yl)methyl]-1,4,9-triazaspiro[5.5]undecan-9-yl}butan-1-one
N-cyclopropyl-N-[(4-methoxyphenyl)methyl]furan-2-carboxamide
6-(3-benzoylpiperidine-1-carbonyl)-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
methyl 9-[(3S,4S)-3-hydroxy-4-(pyrrolidin-1-yl)pyrrolidin-1-yl]-3-azaspiro[5.5]undecane-3-carboxylate
1-butyl-3-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidine
N-ethyl-5-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrimidin-2-amine
3-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
3-(2H-1,3-benzodioxol-5-yl)-5-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
1-(4-aminopyrimidin-2-yl)-4-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-1,4-diazepan-6-ol
7-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
8-[(2,6-dimethylphenyl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(4-fluoro-3-methoxyphenyl)-3-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}urea
1-(3-chlorophenyl)-4-[(3-{2-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl]piperazine
1-(1-benzothiophene-5-carbonyl)-3-(3-methoxypropyl)piperidine
2-[1-(2,6-dimethoxypyrimidin-4-yl)piperidin-3-yl]ethan-1-amine
1-[4-({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)piperidin-1-yl]ethan-1-one
3-(5-{[2-(ethylsulfanyl)-1,3-thiazol-4-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridazine
2-{[(1-methyl-1H-imidazol-2-yl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
3-hydroxy-3-({[2-(2-oxoimidazolidin-1-yl)ethyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
(4aS,8aS)-2-{2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}-decahydroisoquinoline
1-{4-[2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
N-{[2-(dimethylamino)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]oxolane-2-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]acetamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl})amine
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-N,N-diethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
methyl 3-cyclobutaneamido-1-[2-(pyridin-2-yl)ethyl]-5-[(4,4,4-trifluorobutan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate