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N-[3-({[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]carbamoyl}methoxy)phenyl]propanamide
1-(2,2-dimethylpropyl)-4-[(2-methyl-5-propylpyrimidin-4-yl)amino]pyrrolidin-2-one
4-(3-benzyl-1H-pyrazol-5-yl)-1-{spiro[2.3]hexane-1-carbonyl}piperidine
{1-[1-(6-methylpyridine-3-carbonyl)piperidin-3-yl]piperidin-4-yl}methanol
3-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-methyl-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-ethyl-4-[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
6-(azepan-1-yl)-N-[3-(morpholin-4-yl)propyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-butyl-8-[(1-methyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[2-(5,6-dimethoxy-1-oxo-1,2-dihydroisoquinolin-2-yl)acetyl]piperidine-3-carbonitrile
2-({cyclopropyl[(3-ethoxyphenyl)methyl]amino}methyl)quinolin-8-ol
4-(1-{[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propyl)phenol
5-[3-(methoxymethyl)piperidine-1-carbonyl]-2-(pyridin-3-yl)pyridine
1-ethyl-N-(furan-2-ylmethyl)-N-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-{4-[(dimethylamino)methyl]-1H-1,2,3-triazol-1-yl}-N-[(1S)-1-phenylethyl]piperidine-1-carboxamide
4-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}phenol
4-[2-(2,2-diphenylethyl)morpholin-4-yl]pyrimidin-2-amine
1-(2-methyl-1,3-benzothiazole-6-carbonyl)azepan-3-amine
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-4-methyl-2-(propan-2-yl)pyrimidine-5-carboxamide
2-[2-(2-methoxyethyl)pyrimidin-5-yl]-7,8-dimethyl-4-(piperidine-1-carbonyl)quinoline
N-{1-[(2,2-difluoro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}methanesulfonamide
N-(pyridin-2-ylmethyl)-4-{[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]oxy}benzamide
2-(1H-1,3-benzodiazol-1-yl)-N-(cyclohex-1-en-1-ylmethyl)propanamide
N-(1,3-benzoxazol-2-ylmethyl)-2-ethyl-N,4-dimethyl-1,3-oxazole-5-carboxamide
1-(oxolan-2-ylmethyl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-(prop-2-en-1-yl)-4-{3-[(pyridin-2-ylmethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxamide
4-[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]-N,N-dimethylpiperazine-1-sulfonamide
[5-({[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amino}methyl)furan-2-yl]methanol
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(quinazolin-4-yloxy)acetamide
N5-[2-(4-chlorophenyl)ethyl]-1-cyclopentyl-N3-methyl-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-[(3,5-dimethoxyphenyl)methyl]-4,5-dimethyl-2,3-dihydro-1,3-oxazol-2-one
3,5-dimethyl-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)-1H-pyrazole-4-sulfonamide
1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(pyridin-2-yl)ethan-1-one
(1S,5R)-6-propyl-3-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]butan-1-one
N-[2,4-dichloro-5-(propan-2-yloxy)phenyl]-4-methoxypiperidine-1-carboxamide
5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-N-[2-(1,3-thiazol-4-yl)ethyl]pyridin-2-amine
3-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-1-[3-(2-oxopyrrolidin-1-yl)phenyl]urea
1-tert-butyl-N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N-methyl-5-oxopyrrolidine-3-carboxamide
5-({[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl]amino}methyl)-N-methyl-1,2,4-oxadiazole-3-carboxamide
(1S,5R)-3-(5-fluoropyridine-3-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,2,2-trimethyloxane-4-carboxamide
(1R,3S)-3-[1-butyl-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]cyclopentan-1-amine
2-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]pyridine-4-carbonitrile
N-benzyl-2-[2-(2-hydroxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]propanamide
N-ethyl-N-(pyridin-4-ylmethyl)-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
6-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,3-benzothiazole
2-[({3-[2-(dimethylamino)acetamido]phenyl}carbamoyl)amino]-N,N-dimethylacetamide
4-{2-[(1-benzylpyrrolidin-3-yl)carbamoyl]ethyl}-N-(propan-2-yl)piperidine-1-carboxamide