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2-{1-ethyl-8-[(3-methoxyphenyl)methyl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
(1S,5R)-3-methyl-6-[4-(trifluoromethyl)benzenesulfonyl]-3,6-diazabicyclo[3.2.2]nonane
3-[(1-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methyl]benzoic acid
2-{[(2,3-dimethyl-1H-indol-5-yl)methyl]amino}-6-methylpyridine-3-carboxamide
(4aR,8aR)-4-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-2H-1,4-benzoxazine
1-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}cyclopropan-1-amine
3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-4,5,6,7-tetrahydro-1-benzofuran-4-one
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-3-(4-methylphenoxymethyl)piperidine
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-pyrazol-1-yl)propan-1-one
4-{5-[(methylsulfanyl)methyl]-1-(pyridin-2-yl)-1H-1,2,4-triazol-3-yl}benzamide
3-{1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidin-2-yl}propanoic acid
N-{[3-(dimethylamino)phenyl]methyl}-3-(1H-pyrazol-1-yl)benzamide
2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-5-methoxyphenol
(3R,4R)-1-[(dimethyl-1,3-thiazol-2-yl)methyl]-3,4-dimethylpyrrolidin-3-ol
1-ethyl-3,5-dimethyl-4-({2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-1H-pyrazole
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]acetamide
4-[(2-chloro-6-fluorophenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-[4-(thiomorpholine-4-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]azetidin-3-yl}pyridine
5-(phenoxymethyl)-N-[(2,4,6-trimethylphenyl)methyl]-1H-pyrazole-3-carboxamide
9-[(2S)-2-aminopentanoyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(2,3-dihydroxypropyl)-2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-[(2-fluorophenyl)methyl]piperidine
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-4-oxo-3,4-dihydroquinazoline-2-carboxamide
(3S,4R)-1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
1-[2-(furan-2-yl)-4-(1,4-oxazepan-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[(oxolan-3-yl)amino]pyridine-3-carboxamide
N-{[1-(4-methylpiperazin-1-yl)cyclohexyl]methyl}-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
1-(2,2-dimethylpropyl)-3-hydroxy-3-({[(3-phenyl-1H-pyrazol-4-yl)methyl]amino}methyl)piperidin-2-one
2-{2-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]-2-oxoethyl}-3-phenylcyclopent-2-en-1-one
1-(cyclohex-3-ene-1-carbonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-cyclopentanecarbonyl-N-[4-(3-fluorophenyl)phenyl]piperidine-3-carboxamide
2-(3-fluorophenoxymethyl)-N-[(1R,2S)-2-phenylcyclopropyl]-1,3-oxazole-4-carboxamide
2-(2-{1-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
N-cyclopentyl-1-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
N-[(3R,5S)-5-[(propan-2-yl)carbamoyl]-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
N-[2-(dimethylsulfamoyl)ethyl]-2-(phenylamino)pyrimidine-5-carboxamide
methyl 2-{[3-oxo-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decane-8-carbonyl]amino}acetate
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl][(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]methylamine
N-(2-methoxyethyl)-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}-1,3-thiazole-5-carboxamide
3-hexyl-8-(5-methylpyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,3-dimethylbenzamide
2-fluoro-N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)benzamide
N-{4-[4-(4-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxy)piperidine-1-carbonyl]phenyl}acetamide
5-[2-(aminomethyl)-7-chloro-2,3-dihydro-1-benzofuran-5-yl]-N-propylthiophene-2-carboxamide
4-methyl-2-(propan-2-yl)-N-(2-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1,3-thiazole-5-carboxamide
1-[(3R,5R)-3-(hydroxymethyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-1-yl]-2-(2H-1,2,3-triazol-2-yl)ethan-1-one
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-{[(4-methylphenyl)amino]methyl}benzamide
4-[4-(8-chloroquinolin-2-yl)piperazin-1-yl]quinazoline