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8-cyclopropyl-N-[3-(methylsulfanyl)phenyl]-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
[5-fluoro-7-(1H-indazol-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
1-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-amine
N-cyclopropyl-2-{[(3-hydroxy-2-oxo-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]amino}acetamide
N-({5-[(2,3-difluoro-6-methoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
4-hydroxy-N-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]piperidine-1-carboxamide
N-ethyl-N-(oxan-4-ylmethyl)-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-ethyl-1,6-dimethyl-N-(2-methylprop-2-en-1-yl)-4-oxo-1,4-dihydroquinoline-3-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-N-(furan-2-ylmethyl)-5-methoxybenzamide
1-{4-[(dimethylsulfamoyl)amino]phenyl}-N-(1H-indol-2-ylmethyl)piperidin-4-amine
6-(benzyloxy)-4-(5-methyl-1H-pyrazole-3-carbonyl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-1-[2-(trifluoromethyl)pyrrolidin-1-yl]propan-1-one
2-[(3aS,6aR)-3-cyclopentyl-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]-6-methylpyridine-3-carboxamide
3-{2-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
1-[3-(1H-pyrazol-1-yl)benzoyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
(3S,9aR)-8-[(3-fluoro-4-methylphenyl)methyl]-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-({2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)pyridine-3-carboxylic acid
ethyl 1-(2,2-diphenylethyl)-4-(2-methoxyethyl)piperidine-4-carboxylate
N-{4-[4-({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)piperidin-1-yl]phenyl}-2-phenoxyacetamide
9-(but-3-yn-1-yloxy)-4-(2-methyl-1,3-thiazole-4-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[3-(1-phenylcyclopropyl)-5-(propoxymethyl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
(3S,4S)-4-methyl-1-(1,2,3,4-tetrahydroquinoline-8-carbonyl)piperidine-3,4-diol
3-{[2-(1-methyl-1H-pyrazol-5-yl)ethyl]sulfamoyl}-N-(pyrrolidin-3-yl)benzamide
N-[1-(4-fluorophenyl)-2-hydroxyethyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
N-[3-(azepan-1-yl)propyl]-N-methyl-3-(1H-pyrazol-4-yl)benzamide
N,1-dimethyl-N-{2-phenyl-1-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-4-yl]ethyl}-1H-pyrazole-3-carboxamide
6-(4-methoxyphenyl)-9-(3-methylthiophene-2-carbonyl)-6,9-diazaspiro[4.5]decan-7-one
1-(azocan-1-yl)-3-(2-methoxy-4-{[4-(methoxymethyl)piperidin-1-yl]methyl}phenoxy)propan-2-ol
3,5-dichloro-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}pyridin-2-amine
(2S)-2-[(4-{[(1-methyl-1H-pyrazol-4-yl)methyl]sulfamoyl}phenyl)formamido]propanamide
1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3-[2-(4-fluorophenyl)ethyl]piperidine
3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-3-yl}-N-[(2-chlorophenyl)methyl]propanamide
N-(2,4-dimethoxyphenyl)-3-[1-(2-methoxy-2-phenylacetyl)piperidin-4-yl]propanamide
N-cyclopropyl-2-[4-(4-methoxyphenoxy)piperidin-1-yl]pyridine-4-carboxamide
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(naphthalen-2-yloxy)ethan-1-one
3-ethoxy-1-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
2-ethyl-8-(5-methylpyrazine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-2,4-dimethyl-1,3-thiazole-5-carboxamide
[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({3-methoxy-2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)amine
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-ethyl-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
3-(5-cyclobutyl-1,3,4-thiadiazol-2-yl)-1-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}urea
1-(1H-imidazol-2-ylmethyl)-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
(2R,6R)-11-methoxy-4-(2-methoxyethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-(2,5-dimethylphenyl)-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
2-[3-(pyridin-4-yl)azetidin-1-yl]-6-(trifluoromethyl)pyridine
2-(4-methoxy-2-methylphenyl)-2-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]acetic acid
2-(3-fluorophenyl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
(2E)-3-(1-methyl-1H-pyrazol-4-yl)-1-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}prop-2-en-1-one
(2S,4R)-4-amino-N-methyl-1-[(6-phenoxypyridin-3-yl)methyl]pyrrolidine-2-carboxamide
7-methoxy-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide