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3-(2-methyl-1H-1,3-benzodiazol-1-yl)-1-[3-(pyridin-2-yl)azetidin-1-yl]propan-1-one
6-chloro-2-{1-[5-(5-methylfuran-2-yl)-1,2,4-triazin-3-yl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
(1R,3S)-N3-ethyl-1,2,2-trimethyl-N1-[(5-methylpyrazin-2-yl)methyl]cyclopentane-1,3-dicarboxamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-1,3-benzothiazole-2-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-3,5-dimethyl-1H-pyrazol-1-yl]-N-(1,3-dimethyl-1H-pyrazol-5-yl)acetamide
[(3-{[1-(2-cyclopropylquinoline-4-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(thiophen-2-ylmethyl)amine
3-phenyl-1-[4-(1H-1,2,4-triazol-1-yl)butyl]pyrrolidin-3-ol
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(4-methoxyphenyl)-4-oxobutanamide
5-[4-(1H-imidazol-1-yl)phenoxymethyl]-3-propyl-1,2,4-oxadiazole
2-amino-4-[2-methoxy-5-(propan-2-yl)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-(dimethylamino)-2-(3-methylphenyl)-N-[(1r,4r)-4-hydroxycyclohexyl]acetamide
1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}-3-(pyrazin-2-yl)propan-1-one
1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-propoxypiperidine
2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-(pyridin-3-yl)ethan-1-ol
N-(4-methoxyphenyl)-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-amine
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-(2-ethyl-1H-imidazol-1-yl)acetamide
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methylcyclopropane-1-carboxamide
N,1-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
2-(4-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperazin-1-yl)pyrazine
N-cyclopropyl-1-(1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
3-(1-{[6-(dimethylamino)pyridin-3-yl]methyl}piperidin-3-yl)benzoic acid
4-(2-methylpropyl)-1-(2-phenoxypropanoyl)-1,4-diazepan-5-one
ethyl 3,5-dimethyl-4-{[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]carbamoyl}-1H-pyrrole-2-carboxylate
2-(1-{[1-(3-methyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
1-(carbamoylmethyl)-N-[2-(dimethylamino)-2-(4-fluorophenyl)ethyl]piperidine-4-carboxamide
1-cyclohexyl-4-[3-(pyrrolidin-1-ylmethyl)imidazo[1,2-a]pyridine-2-carbonyl]piperazine
(2S)-2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-(2,4-dichloro-5-fluorophenyl)pyrrolidine-1-carboxamide
2-oxo-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(pyrrolidin-1-yl)acetamide
N-[(5-methylpyrazin-2-yl)methyl]-4-(pyridin-4-yl)pyrimidin-2-amine
2-methyl-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrido[2,3-d]pyrimidin-4-amine
2-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidine-1-carbonyl]benzonitrile
6,7-dimethoxy-3-[(5-methylthiophen-2-yl)methyl]-3,4-dihydroquinazolin-4-one
(1S,5R)-3-cyclobutanecarbonyl-6-(3-propyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(2S,4S)-4-amino-N-ethyl-1-{2-[(4-ethylcyclohexyl)formamido]acetyl}pyrrolidine-2-carboxamide
1-(5-{[4-(2-hydroxyethyl)piperidin-1-yl]methyl}-2-methoxyphenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidine
2-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-(2-oxo-2-{2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
2-[(cyclopropylmethyl)sulfanyl]-1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
3-[1-(1-benzothiophen-5-ylmethyl)-1H-1,2,3-triazol-4-yl]phenol
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-pyrrol-1-yl)butan-1-one
4-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]azetidin-3-yl}morpholine
N-[4-(1H-pyrazol-5-yl)phenyl]-1-(thiophen-3-ylmethyl)piperidine-3-carboxamide
2-(2,3-dihydro-1H-isoindole-2-carbonyl)-5-methoxy-1-methyl-1H-indole
1-[(2,3-difluorophenyl)methyl]-3-{[(hexahydro-1H-pyrrolizin-7a-ylmethyl)amino]methyl}-3-hydroxypiperidin-2-one
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
3-{4-[4-(pyridin-2-yl)pyrimidin-2-yl]piperazin-1-yl}-1-azabicyclo[2.2.2]octane
[(5-methylfuran-2-yl)methyl]({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)amine