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N-[(1-benzyl-1H-imidazol-2-yl)methyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-[4-(dimethylamino)azepan-1-yl]-2-(4-phenylphenyl)ethan-1-one
N-[(2-hydroxyphenyl)methyl]-N-methyl-2-(4-propanoylphenoxy)acetamide
4-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]propan-1-one
2-ethoxy-5-{2-[(1-methylpiperidin-3-yl)amino]pyrimidin-4-yl}benzoic acid
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-(pyridin-3-ylmethyl)-2-(pyridin-3-yloxy)acetamide
3-[(1R,3R)-3-aminocyclopentyl]-1-(3-chloro-4-methoxyphenyl)urea
2-methyl-5-(2-{2-[(quinolin-2-yl)amino]ethyl}morpholin-4-yl)-2,3-dihydropyridazin-3-one
4-[2-(3-hydroxypropyl)-1H-1,3-benzodiazol-1-yl]-2-(1,2-oxazol-5-yl)phenol
8-[(4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]quinoline
3-(5-methylthiophen-2-yl)-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
5-acetyl-N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide
N-[(4,6-dimethylpyridin-3-yl)methyl]-2-(1-ethylpiperidin-4-yl)acetamide
2-methoxy-6-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(1,3-thiazol-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(3-methylpyridin-2-yl)methyl]-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
[(2S)-1-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}pyrrolidin-2-yl]methanol
2-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]-N-[5-(methoxymethyl)-1,3,4-thiadiazol-2-yl]acetamide
1-[4-(7-{[4-(benzyloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)piperidin-1-yl]ethan-1-one
methyl 2-(ethylsulfamoyl)-6-(4-phenylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}-1H-indole
(3aS,6aR)-5-{[2-(furan-2-yl)phenyl]methyl}-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(2R)-2-(methoxymethyl)-N-[2-(2-phenoxyethoxy)phenyl]pyrrolidine-1-carboxamide
N3-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
3-ethyl-1-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidin-3-ol
4-{4-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]piperidin-1-yl}-5-propylpyrimidine
N-(4-{1-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}phenyl)acetamide
1-methyl-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]azepane-2-carboxamide
{1-cyclopentanecarbonyl-3-[(2-methylphenyl)methyl]piperidin-3-yl}methanol
2-(phenylamino)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)pyrimidine-5-carboxamide
methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})(thiophen-2-ylmethyl)amine
1-(benzyloxy)-8-[2-(3-phenyl-1H-1,2,4-triazol-5-yl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
1-[4-(3-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}phenoxy)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
1-(cyclopropylmethyl)-3-(2,3-dimethoxyphenyl)-6-(1H-imidazol-2-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N,N-dimethyl-3-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}pyrazin-2-amine
N-methyl-N-(pyridin-2-ylmethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N,N-dimethyl-4-[2-(2-phenylethyl)morpholine-4-carbonyl]piperidine-1-carboxamide
1-(4-pentanamidobenzoyl)piperidine-2-carboxylic acid
2-benzyl-8-(3-ethyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
3-chloro-5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridin-2-one
2-[3-fluoro-5-(2-methylpropoxy)phenyl]-N-(propan-2-yl)pyridine-4-carboxamide
3-[2-oxo-2-(5-oxo-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-1-yl)ethyl]-2,3-dihydro-1H-isoindol-1-one
1-benzyl-N,N-dimethyl-5-{[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]pyrimidin-4-amine
2-[4-(furan-2-yl)phenyl]-1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazole
1-[2-(6-methylpyridin-2-yl)ethyl]-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
[1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)pyrrolidin-3-yl]methanamine
(2S,4S)-4-[(2,3-dihydro-1H-inden-2-yl)amino]-1-[(2E)-3-phenylprop-2-en-1-yl]-N-(propan-2-yl)pyrrolidine-2-carboxamide