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1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-(2-methylprop-2-en-1-yl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
4-[(benzyloxy)methyl]-1-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-1,2,3-triazole
N-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-(2-fluorophenyl)piperidin-4-amine
4-(4-{[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}piperidin-1-yl)-N-(pyridin-3-ylmethyl)benzamide
[(3R,4R)-1-(1H-1,3-benzodiazol-2-ylmethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-[3-(dimethylamino)-2,2-dimethylpropyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
4-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-6-methyl-1,2-dihydroquinolin-2-one
1-{2-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
N-{3-methyl-1-[7-(5-phenoxyfuran-2-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}acetamide
N2-cyclopropyl-N4-[2-(6-methylpyridin-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-{2-[(pyridin-3-yl)amino]ethyl}-1H-1,3-benzodiazole-2-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-N'-(2-ethoxyphenyl)propanediamide
5-[(2E)-but-2-en-2-yl]-1-[3-(1H-imidazol-1-yl)propyl]-4-phenyl-1H-imidazole
(1S,5R)-N-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carboxamide
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](methyl)[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amine
1-methanesulfonyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)pyrrolidine-2-carboxamide
2-{[3-(1,4-diazepan-1-ylmethyl)-6-methoxyquinolin-2-yl]sulfanyl}acetic acid
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
1-[(4-methylpiperazin-1-yl)sulfonyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
3-cyclopropyl-1-methyl-4-[2-(2-methylphenyl)-1,3-thiazol-5-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-(2H-1,3-benzodioxol-4-ylmethyl)-6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
(3-{2-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
N'-[2-(2,4-dimethylphenoxy)ethyl]-N'-methylpentanediamide
N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
ethyl 1-(dimethylsulfamoyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
3-({2-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
N-(3,5-dimethylphenyl)-6-propanoyl-6-azaspiro[2.5]octane-1-carboxamide
3-{2-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-1H-pyrrol-1-yl}pyridine
3-hydroxy-S-[2-(3,3,3-trifluoropropanoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]butane-1-sulfonamido
2-methoxy-4,6-dimethyl-5-[3-(morpholin-4-ylmethyl)phenyl]pyridine-3-carbonitrile
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(adamantan-1-ylmethyl)({[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl})methylamine
(3S,4R)-1-(4-methanesulfonylbenzoyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
(3R,4R)-3-cyclobutyl-4-methyl-1-(2-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-3-ol
1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}ethan-1-one
6-[2-(4-fluorophenoxy)ethyl]-2-methyl-[1,2,4]triazolo[1,5-a]pyridine
ethyl 4-{[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]amino}piperidine-1-carboxylate
N-[2-(2-chlorophenyl)ethyl]-3-(morpholine-4-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
(4aS,7aR)-1-(4-methyl-1H-imidazole-5-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methyl-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
1-[(1R,5R)-6-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-ethyl-6-methyl-3-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
1-(3-methoxypyrazin-2-yl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
1-[(4aR,8aR)-7-[(2-chlorophenyl)methyl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
N-(2,3-dihydro-1H-inden-2-yl)-N,2-dimethyl-1,3-thiazole-4-carboxamide
2-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-4-oxo-4,5,6,7-tetrahydro-1H-indole-3-carboxamide