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1-tert-butyl-5-cyclobutyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
3-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)-4,6-dimethyl-1,2-dihydropyridin-2-one
1-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
8-methoxy-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1,4-oxazepan-6-ol
2-({3-oxo-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-9-yl}methyl)benzonitrile
N-(6-fluoropyridin-3-yl)-4-(2-methoxyacetyl)-1,4-diazepane-1-carboxamide
1-(furan-3-carbonyl)-4-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1,4-diazepan-6-ol
2-butyl-8-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-4-propyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1,2,3-thiadiazole-5-carboxamide
2-[(4-aminoazepan-1-yl)methyl]-5,8-dimethylquinolin-4-ol
(3S,4R)-3-methoxy-1-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}piperidin-4-amine
2-[4-(2-amino-6-methoxypyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-ethyl-1H-1,2,3-triazol-4-yl)acetamide
1-ethyl-3-(thiomorpholine-4-carbonyl)-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(2-fluoro-5-methylphenoxy)-1-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]piperidine-4-carboxylic acid
{[4-(3,6-dimethyl-1-benzofuran-2-carbonyl)-1,4-oxazepan-6-yl]methyl}dimethylamine
4-({5-[1-(3-fluoropyridin-2-yl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
(1S,5R)-6-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-hydroxy-2-(pyridin-2-yl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(3S)-1-benzylpyrrolidin-3-yl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propanamide
N-[(5-chlorothiophen-2-yl)methyl]-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
1-methanesulfonyl-N-methyl-N-[(3-methylpyridin-4-yl)methyl]pyrrolidine-2-carboxamide
(4aS,8aS)-2-(5-fluoro-4-methoxypyrimidin-2-yl)-decahydro-2,7-naphthyridin-4a-ol
2-[({[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}amino)methyl]-6-methylquinolin-4-ol
3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}-N-ethylpyrrolidine-1-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-1,1-dioxo-N-propyl-1λ6-thiolane-3-carboxamide
[2-propoxy-5-(pyridin-3-yl)phenyl]methanol
8-[1-(methoxymethyl)cyclobutanecarbonyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-methyl-6-(1-methyl-1H-imidazol-2-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)pyridazin-3-amine
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)piperidin-2-one
8-[(3E)-pent-3-enoyl]-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1,3-thiazol-4-yl)ethyl]acetamide
3-(3-cyclohexyl-1H-1,2,4-triazol-5-yl)-1-[(4-methylphenyl)methyl]urea
1-methyl-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}piperidine-2-carboxamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(1-ethyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[(8-methoxyquinolin-2-yl)amino]acetamide
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-1-methanesulfonylpiperidin-4-amine
2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]-N,N-dipropylacetamide
4-(2-fluorophenoxy)-1-(thiophene-3-carbonyl)piperidine-4-carboxylic acid
(3S,4R)-1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
3-(2-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)-2,3-dihydro-1λ6-thiophene-1,1-dione
2-(4-{1-butyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-2-chlorophenoxy)acetamide
4-(2,6-dimethylpyridin-3-yl)-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]pyrimidin-2-amine
1-[2-methoxy-5-({[3-(pyridin-3-yloxy)propyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
3-(1-methylpiperidin-3-yl)-N-[2-(pyrazin-2-yl)ethyl]propanamide
5-cyclopropyl-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
N,2-dimethyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-6-(piperidin-3-yl)pyrimidin-4-amine
(3R,4R)-1-[3-(4-fluorophenyl)benzoyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
ethyl N-(4-cyclopentyl-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)carbamate