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N-(1-benzylpiperidin-4-yl)-2-cyclopropyl-1-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-2-[3-(methylsulfanyl)phenyl]ethan-1-one
4-[1-(4-methoxy-2-methylphenyl)-1H-imidazol-2-yl]pyridine
8-[5-(1H-imidazol-2-yl)thiophene-2-carbonyl]-2-methyl-2,8-diazaspiro[4.5]decane
(2R,6R)-11-methoxy-4-(pyridin-4-ylmethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-methyl-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-1H-1,3-benzodiazole-5-carboxamide
(1S,5R)-6-[(3,5-difluorophenyl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-[({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)(methyl)amino]-1λ6-thiolane-1,1-dione
1-[(2-fluorophenyl)methyl]-6-oxo-N-{[4-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidine-3-carboxamide
4-[(3-fluorophenyl)methyl]-3-[3-(morpholin-4-yl)propyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
6-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
8-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}pyrazolo[1,5-a]pyridine-3-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-[(1,2-oxazol-3-ylmethyl)sulfamoyl]benzamide
4-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
methyl 3-{[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetamido]methyl}-5-[(2E)-3-phenylprop-2-enamido]benzoate
N-(2-methoxyethyl)-2-(pyridin-4-yl)-N-(1,3-thiazol-2-ylmethyl)pyrimidine-5-carboxamide
1-[(3-methoxyphenyl)methyl]-5-{2-[(pyridin-2-ylmethyl)amino]ethyl}pyrrolidin-2-one
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[2-(dimethylamino)acetyl]pyrrolidine-3-carboxylic acid
5-methoxy-1-methyl-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-1H-indole-2-carboxamide
2-methyl-N-{2-[7-(5-phenoxyfuran-2-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}propanamide
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
7-(5-fluoro-2-methylbenzoyl)-N,N-dimethyl-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-[1-(propan-2-yl)-1H-pyrazol-5-yl]urea
2-(3-hydroxypropyl)-8-(9H-purin-6-yl)-2,8-diazaspiro[5.5]undecan-3-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-{2-[methyl(phenyl)amino]propyl}propanamide
N-[2-(5-methylfuran-2-yl)ethyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
1-{5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-yl}piperidin-4-ol
N-(5-{[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]sulfonyl}-1,3-thiazol-2-yl)acetamide
(3aR,6aR)-2-methanesulfonyl-5-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-({1-[(1-{furo[3,2-c]pyridin-4-yl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)piperazin-2-one
4-[2-(morpholin-4-yl)-2-oxoethyl]-N-(2-propylphenyl)piperazine-1-carboxamide
[5-({3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}methyl)-2-ethoxyphenyl]methanol
N-(2-hydroxyethyl)-1-[1-(isoquinolin-1-yl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
1-(2-methylpyridin-4-yl)-4-(6-phenylpyridazin-3-yl)-1,4-diazepane
(1S,3R)-N1-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
1-cyclopentyl-5-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]piperidin-2-one
1-[2-(1H-indol-3-yl)ethyl]-3-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]urea
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one
1-(prop-2-en-1-yl)-4-(3-propyl-1H-pyrazole-5-carbonyl)piperazine
(2S,4R)-4-amino-N,N-diethyl-1-(3-oxo-3,4-dihydroquinoxaline-2-carbonyl)pyrrolidine-2-carboxamide
7-methyl-2-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
1-(2-fluorophenyl)-2-(furan-3-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
methyl (2S)-2-[3-(2-ethyl-5-oxopyrrolidin-2-yl)propanamido]-2-phenylacetate
N-ethyl-5-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2,6-dioxo-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
7-methyl-2-[2-(5-oxo-2-phenylcyclopent-1-en-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-{2-[(3-ethenylphenyl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}-3-methoxypropan-1-one
5-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
N-[(3S,4R)-1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-4-propylpyrrolidin-3-yl]acetamide