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1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-2-hydroxy-4-(methylsulfanyl)butan-1-one
methyl 4-[3-cyclopropyl-1-(6-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]butanoate
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-(4-methylphenyl)cyclopropane-1-carboxamide
1-(4-methyl-2-{[2-(pyrrolidin-1-yl)ethyl]amino}pyrimidin-5-yl)ethan-1-one
3-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]pyridin-2-ol
methyl 1-(2-methoxyethyl)-5-{[(2E)-2-methylbut-2-en-1-yl]amino}-3-(3-methylbutanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(3R,5S)-1-benzyl-5-(3-fluorophenoxymethyl)-N-(3-methoxypropyl)piperidine-3-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(4-methyl-2-oxo-2H-chromen-7-yl)azetidine-1-carboxamide
2-(4-fluorophenoxymethyl)-N-methyl-N-(propan-2-yl)-1,3-oxazole-4-carboxamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(6-methyl-2-propylpyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-phenoxypiperidine-4-carboxylic acid
2-[1-ethyl-2,4-dioxo-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
3-(2-methoxyphenoxy)-1-(7-methyl-1-benzofuran-2-carbonyl)azetidine
N,6-dimethyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-(2-methoxyethyl)-1-[(2,4,5-trimethylphenyl)methyl]-1,4-diazepan-5-one
2-benzyl-8-[5-(methoxymethyl)furan-2-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
5-{[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]methyl}-2-(thiophen-2-yl)pyrimidine
ethyl 1-(3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}propanoyl)piperidine-4-carboxylate
2-{5-[(3-hydroxyphenyl)methyl]-3-(2-methoxyethyl)-1H-1,2,4-triazol-1-yl}benzoic acid
1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(1H-pyrazol-4-yl)propan-1-one
2-[cyclopentyl(methyl)amino]-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
N-(6-methylpyridin-3-yl)quinoxaline-6-carboxamide
(1S,5R)-3-[2-(3,4-dimethylphenoxy)ethyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
(2S,4S)-4-amino-N,N-diethyl-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]pyrrolidine-2-carboxamide
ethyl[(1-methyl-1H-imidazol-2-yl)methyl]{[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine
3-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-N-[2-(dimethylamino)ethyl]propanamide
{1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]pyrrolidin-3-yl}methanamine
3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
N-benzyl-5-methyl-N-[(6-methylpyridin-2-yl)methyl]-1,3,4-oxadiazole-2-carboxamide
N-(1-{4-[(cyclopropylmethyl)(oxolan-2-ylmethyl)carbamoyl]phenyl}-1H-pyrazol-4-yl)-2,4-dimethylbenzamide
2,6-dimethyl-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]quinoline-4-carboxamide
2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]-N-(2-phenoxyethyl)acetamide
(3R,4S)-1-(1-ethyl-1H-pyrazole-4-carbonyl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
N-ethyl-N-(pyridin-4-ylmethyl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-amine
4-methoxy-2-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]phenol
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-(1-methoxybutan-2-yl)benzamide
2-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]pyridine-3-carbonitrile
N-cyclopropyl-4-fluoro-N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)benzamide
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]piperidin-4-amine
dimethyl({4-[1-(thiophene-2-carbonyl)piperidin-2-yl]phenyl}methyl)amine
N,2-dimethyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}imidazo[1,2-a]pyrimidine-3-carboxamide
3-(4-ethoxyphenyl)-3-[(2-oxo-1,2-dihydroquinolin-4-yl)formamido]propanoic acid
1-[(2-chloro-4-fluorophenyl)methyl]-N-[3-(methylsulfanyl)propyl]-1H-1,2,3-triazole-4-carboxamide
3-(azepane-1-carbonyl)-1-ethyl-N-[2-(3-methoxyphenyl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-chloro-N-[(3R,4S)-1-[(methylcarbamoyl)methyl]-4-propylpyrrolidin-3-yl]thiophene-2-carboxamide
N-{2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
4-(piperidin-1-yl)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}butan-1-one
(3S,4R)-1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
(5-{1-[(5-ethylpyridin-2-yl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide