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2-tert-butyl-4-hydroxy-N-[2-(4-phenylpiperidin-1-yl)ethyl]pyrimidine-5-carboxamide
N-[1-(3-methylpyridin-2-yl)propyl]-6-(piperidin-1-yl)pyrimidin-4-amine
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperidine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-[3-(methylsulfanyl)propanoyl]-1,4-diazepan-2-one
1,5-dimethyl-3-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1H-indazole
2-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-4-phenyl-1,3-thiazole
2-cyclopropanecarbonyl-8-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
ethyl 2-{3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-methylpropanamido}acetate
1-{1-methyl-5-[(2-{[methyl(propyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)methyl]-1H-pyrrol-3-yl}ethan-1-one
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carboxamide
4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethyl]pyrimidin-2-amine
2-(2-hydroxyethyl)-9-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{3-[4-({[(4-fluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
N4-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-5,6-dimethylpyrimidine-2,4-diamine
2-(3-acetyl-4-methoxyphenyl)benzamide
7-[(2,3-difluorophenyl)methyl]-2-(2-methylpropyl)-2,7-diazaspiro[4.5]decan-6-one
1-[3-(furan-2-yl)phenyl]-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}piperidin-4-amine
7-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-3H,4H,5H-pyridazino[4,5-b]indol-4-one
4-({2-[3-(azepan-1-yl)-2-hydroxypropoxy]-5-chlorophenyl}methyl)piperazine-1-carbaldehyde
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[(4-fluorophenyl)formamido]propanamide
N,2-dimethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-(1-methoxypropan-2-yl)-5-methyl-4-[(2-phenylethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2-{1-benzyl-4-[(5-chloro-2,3-dimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
5-(1-butyl-3-methyl-1H-1,2,4-triazol-5-yl)-1-methyl-1,2-dihydropyridin-2-one
[(3R,4R)-1-(5-chloro-2-fluorobenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
(1S,9aR)-1-{[4-(4-methoxybenzoyl)piperazin-1-yl]methyl}-octahydro-1H-quinolizine
2-hydroxy-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)pyridine-3-carboxamide
N-cyclopropyl-2-fluoro-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzamide
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-[(2S)-pyrrolidin-2-ylmethyl]piperidine-4-carboxamide
9-methyl-3-[3-(piperazin-1-yl)propanoyl]-3,9-diazaspiro[5.6]dodecan-10-one
methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)(2-phenylpropyl)amine
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-3-(2-oxopyrrolidin-1-yl)propanamide
1-(4-fluorophenyl)-N-[3-(2-methoxyphenyl)propyl]cyclopropane-1-carboxamide
{[2-(butan-2-ylsulfanyl)pyrimidin-5-yl]methyl}[2-(1H-imidazol-1-yl)ethyl]methylamine
5-(methoxymethyl)-N-({7-[(3-phenoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)furan-2-carboxamide
8-[2-(pyridin-3-yl)-1,3-thiazole-4-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
N-[2-(morpholin-4-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-{[2-(methoxymethyl)-4-methyl-1,3-thiazol-5-yl]methyl}-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
4-(1-phenylethyl)-3-(2-phenylethyl)-4H-1,2,4-triazole
N-[(3R,4S)-1-(cyclobutylmethyl)-4-propylpyrrolidin-3-yl]oxane-4-carboxamide
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-2-oxopiperidin-1-yl]-N,N-dimethylpropanamide
2-(4-{[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]methyl}phenyl)acetic acid
5-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyrazin-2-ol
N-(5-methyl-1,3,4-thiadiazol-2-yl)-2-(oxolane-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
propan-2-yl 2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxylate
N-{1-[4-(3-chlorophenyl)-3-oxopiperazin-1-yl]-3-methyl-1-oxobutan-2-yl}acetamide
(2-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}quinolin-3-yl)methanol
8-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-ethyl-1-(oxan-4-ylmethyl)-3-[4-(trifluoromethyl)phenyl]urea