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{5-[4-(3,4-diethoxyphenyl)-1H-imidazol-2-yl]furan-2-yl}methanol
3-[(3R,4S)-4-(dimethylamino)-1-({1-[4-(propan-2-yl)phenyl]-1H-pyrazol-4-yl}methyl)piperidin-3-yl]propanoic acid
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-[methyl(1-methylpyrrolidin-3-yl)amino]propanamide
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-ethyl-4-{[(3-methylphenyl)methyl]amino}pyrrolidine-2-carboxamide
4-[({2-cyclopentyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)methyl]-1-methylpiperidin-4-ol
6-(3-chlorophenyl)-N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
5-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-1,2-dihydropyridin-2-one
4-ethyl-3-(1-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2R)-1-(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzoyl)pyrrolidine-2-carboxamide
5-(2,6-dimethoxypyridin-3-yl)-N-methyl-4-(4-methylphenyl)pyrimidin-2-amine
2-(3-methoxypropyl)-8-(3-methyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-4-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1-(2-methylpropyl)piperidin-4-amine
1-[benzyl(methyl)amino]-3-(5-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-2-methoxyphenoxy)propan-2-ol
1-tert-butyl-N-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-5-oxopyrrolidine-3-carboxamide
2-[4-(2-methoxyethoxy)phenyl]-N-methylpyrimidin-4-amine
N-[3,3-dimethyl-1-(pyridin-3-yl)butyl]-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
7-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
6-[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]pyrazine-2-carboxamide
1-(4-cyclopentyl-1,4-diazepan-1-yl)-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}ethan-1-one
1-(2-aminopyridine-4-carbonyl)-N,N-dimethylazepan-4-amine
3-[(furan-2-ylmethyl)amino]-N-[3-(1H-imidazol-1-yl)propyl]-5-(pyrrolidine-1-sulfonyl)benzamide
1'-(1-methyl-1H-pyrrole-2-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[1-(thiophen-3-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
5,6-dimethyl-N-{2-[methyl(phenyl)amino]propyl}pyrimidin-4-amine
2-[3-(pyridin-4-yl)-5-[(2,3,4-trifluorophenyl)methyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
2-(2-{5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-phenyl-1H-imidazol-1-yl}ethyl)pyridine
3-phenyl-5-(thiolan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(6-chloro-2-methylpyridin-3-yl)-3-(2-ethylphenoxy)azetidine-1-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[4-(2-ethoxyphenyl)piperazin-1-yl]ethan-1-one
N-(butan-2-yl)-6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-3-(thiophen-3-yl)propanamide
3-{2-oxo-2-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethyl}imidazolidine-2,4-dione
5-(2-cyclopentylacetamido)-N,1-dimethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}acetamide
2,6-dihydroxy-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
4-[1-(2-hydroxyethyl)-5-[3-(pyrrolidin-1-yl)propyl]-1H-1,2,4-triazol-3-yl]phenol
methyl 6-(3,5-difluorobenzoyl)-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]butanamide
2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-3-carbonitrile
3,5-dichloro-4-methyl-N-(5-oxo-1-propylpyrrolidin-3-yl)benzamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-3-(4H-1,2,4-triazol-4-yl)benzamide
(2S,4S)-4-amino-N-(propan-2-yl)-1-(propane-2-sulfonyl)pyrrolidine-2-carboxamide
2-(1-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane-6-carbonyl)-1-methyl-1H-indole
2-[(4-methylphenyl)amino]-2-phenyl-N-(pyridin-2-ylmethyl)propanamide
4-({1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)-1-methylpiperazin-2-one
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2-methoxypyridine-3-carboxamide